[F]FEPPA: Improved Automated Radiosynthesis, Binding Affinity, and Preliminary in Vitro Evaluation in Colorectal Cancer (Q62862505)

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20 March 2020

title

[18F]FEPPA: Improved Automated Radiosynthesis, Binding Affinity, and Preliminary in Vitro Evaluation in Colorectal Cancer (English)

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20 March 2020

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Neydher Berroterán-Infante

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20 March 2020

Theresa Balber

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20 March 2020

Markus Mitterhauser

7

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20 March 2020

Wolfgang Wadsak

8

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20 March 2020

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Marcus Hacker

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20 March 2020

author name string

Petra Fürlinger

3

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Michael Bergmann

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Rupert Lanzenberger

5

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20 March 2020

language of work or name

English

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publication date

21 February 2018

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ACS Medicinal Chemistry Letters

20 March 2020

published in

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volume

9

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issue

3

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page(s)

177-181

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Increase in peripheral benzodiazepine binding sites in colonic adenocarcinoma.

20 March 2020

cites work

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12 December 2020

Dramatic increase in peripheral benzodiazepine binding sites in human colonic adenocarcinoma as compared to normal colon

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12 December 2020

Expression of peripheral benzodiazepine receptor (PBR) in human tumors: relationship to breast, colorectal, and prostate tumor progression

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12 December 2020

Translocator protein (18kDa): new nomenclature for the peripheral-type benzodiazepine receptor based on its structure and molecular function

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12 December 2020

Translocator protein (18 kDa) ligand PK 11195 induces transient mitochondrial Ca2 release leading to transepithelial Cl- secretion in HT-29 human colon cancer cells

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12 December 2020

Synthesis and evaluation in monkey of two sensitive 11C-labeled aryloxyanilide ligands for imaging brain peripheral benzodiazepine receptors in vivo

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12 December 2020

Radiosynthesis and initial evaluation of [18F]-FEPPA for PET imaging of peripheral benzodiazepine receptors

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12 December 2020

Translocator protein (18 kDa) (TSPO) as a therapeutic target for neurological and psychiatric disorders

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12 December 2020

Mixed-affinity binding in humans with 18-kDa translocator protein ligands

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12 December 2020

Biodistribution and radiation dosimetry of the 18 kDa translocator protein (TSPO) radioligand [18F]FEDAA1106: a human whole-body PET study

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12 December 2020

An 18-kDa translocator protein (TSPO) polymorphism explains differences in binding affinity of the PET radioligand PBR28

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12 December 2020

Translocator protein (TSPO) in breast cancer.

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12 December 2020

Translocator protein (18 kDa) polymorphism (rs6971) explains in-vivo brain binding affinity of the PET radioligand [(18)F]-FEPPA.

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12 December 2020

Positron-emission tomography imaging of the TSPO with [(18)F]FEPPA in a preclinical breast cancer model.

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12 December 2020

The translocator protein (TSPO) ligand PK11195 induces apoptosis and cell cycle arrest and sensitizes to chemotherapy treatment in pre- and post-relapse neuroblastoma cell lines

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12 December 2020

[18F]DPA-714: direct comparison with [11C]PK11195 in a model of cerebral ischemia in rats

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12 December 2020

Longitudinal PET imaging of muscular inflammation using 18F-DPA-714 and 18F-Alfatide II and differentiation with tumors

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12 December 2020

Inducible loss of one Apc allele in Lrig1-expressing progenitor cells results in multiple distal colonic tumors with features of familial adenomatous polyposis.

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12 December 2020

In vivo evaluation of inflammatory bowel disease with the aid of μPET and the translocator protein 18 kDa radioligand [18F]DPA-714

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12 December 2020

Facile synthesis of SSR180575 and discovery of 7-chloro-N,N,5-trimethyl-4-oxo-3(6-[(18)F]fluoropyridin-2-yl)-3,5-dihydro-4H-pyridazino[4,5-b]indole-1-acetamide, a potent pyridazinoindole ligand for PET imaging of TSPO in cancer

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12 December 2020

Role of translocator protein density, a marker of neuroinflammation, in the brain during major depressive episodes.

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12 December 2020

TSPO expression in brain tumours: is TSPO a target for brain tumour imaging?

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12 December 2020

Evaluating [11C]PBR28 PET for Monitoring Gut and Brain Inflammation in a Rat Model of Chemically Induced Colitis.

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12 December 2020

Translocator protein (TSPO) ligands for the diagnosis or treatment of neurodegenerative diseases: a patent review (2010 - 2015; part 2).

1 reference

12 December 2020

Translocator protein (TSPO) ligands for the diagnosis or treatment of neurodegenerative diseases: a patent review (2010-2015; part 1).

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12 December 2020

Evaluation of TSPO PET Ligands [18F]VUIIS1009A and [18F]VUIIS1009B: Tracers for Cancer Imaging

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12 December 2020

New approaches for the reliable in vitro assessment of binding affinity based on high-resolution real-time data acquisition of radioligand-receptor binding kinetics

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12 December 2020

Translocator Protein-18 kDa (TSPO) Positron Emission Tomography (PET) Imaging and Its Clinical Impact in Neurodegenerative Diseases

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12 December 2020

Molecular Targets for PET Imaging of Activated Microglia: The Current Situation and Future Expectations

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12 December 2020

10.1021/ACSMEDCHEMLETT.7B00367

Identifiers

DOI

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20 March 2020

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20 March 2020

PubMed publication ID

29541356

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