Gastroprokinetic properties of the benzimidazolone derivative BIMU 1, an agonist at 5-hydroxytryptamine4 and antagonist at 5-hydroxytryptamine3 receptors (Q48146857)

From Wikidata

Jump to navigation Jump to search

scientific article

Language	Label	Description	Also known as
English	Gastroprokinetic properties of the benzimidazolone derivative BIMU 1, an agonist at 5-hydroxytryptamine4 and antagonist at 5-hydroxytryptamine3 receptors	scientific article

Statements

scholarly article

1 reference

Europe PubMed Central

PubMed publication ID

9 February 2018

http://europepmc.org/abstract/MED/8058105

Gastroprokinetic properties of the benzimidazolone derivative BIMU 1, an agonist at 5-hydroxytryptamine4 and antagonist at 5-hydroxytryptamine3 receptors (English)

1 reference

Europe PubMed Central

PubMed publication ID

9 February 2018

http://europepmc.org/abstract/MED/8058105

author name string

C A Rizzi

1

1 reference

Europe PubMed Central

PubMed publication ID

9 February 2018

http://europepmc.org/abstract/MED/8058105

A Sagrada

2

1 reference

Europe PubMed Central

PubMed publication ID

9 February 2018

http://europepmc.org/abstract/MED/8058105

A Schiavone

3

1 reference

Europe PubMed Central

PubMed publication ID

9 February 2018

http://europepmc.org/abstract/MED/8058105

P Schiantarelli

4

1 reference

Europe PubMed Central

PubMed publication ID

9 February 2018

http://europepmc.org/abstract/MED/8058105

R Cesana

5

1 reference

Europe PubMed Central

PubMed publication ID

9 February 2018

http://europepmc.org/abstract/MED/8058105

G B Schiavi

6

1 reference

Europe PubMed Central

PubMed publication ID

9 February 2018

http://europepmc.org/abstract/MED/8058105

H Ladinsky

7

1 reference

Europe PubMed Central

PubMed publication ID

9 February 2018

http://europepmc.org/abstract/MED/8058105

A Donetti

8

1 reference

Europe PubMed Central

PubMed publication ID

9 February 2018

http://europepmc.org/abstract/MED/8058105

publication date

1 April 1994

1 reference

Europe PubMed Central

PubMed publication ID

9 February 2018

http://europepmc.org/abstract/MED/8058105

Naunyn-Schmiedeberg's Archives of Pharmacology

1 reference

Europe PubMed Central

PubMed publication ID

9 February 2018

http://europepmc.org/abstract/MED/8058105

349

1 reference

Europe PubMed Central

PubMed publication ID

9 February 2018

http://europepmc.org/abstract/MED/8058105

4

1 reference

Europe PubMed Central

PubMed publication ID

9 February 2018

http://europepmc.org/abstract/MED/8058105

338-345

1 reference

Europe PubMed Central

PubMed publication ID

9 February 2018

http://europepmc.org/abstract/MED/8058105

Neuropharmacology of emesis induced by anti-cancer therapy.

1 reference

https://api.crossref.org/works/10.1007/BF00170878

21 January 2018

Functionalized congener approach for the design of novel muscarinic agents. Synthesis and pharmacological evaluation of N-methyl-N-[4-(1-pyrrolidinyl)-2-butynyl] amides.

1 reference

https://api.crossref.org/works/10.1007/BF00170878

21 January 2018

A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding

1 reference

https://api.crossref.org/works/10.1007/BF00170878

21 January 2018

Domperidone. A review of its pharmacological activity, pharmacokinetics and therapeutic efficacy in the symptomatic treatment of chronic dyspepsia and as an antiemetic

1 reference

https://api.crossref.org/works/10.1007/BF00170878

21 January 2018

Pharmacological properties of GR38032F, a novel antagonist at 5-HT3 receptors

1 reference

https://api.crossref.org/works/10.1007/BF00170878

21 January 2018

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

1 reference

https://api.crossref.org/works/10.1007/BF00170878

21 January 2018

The effect of GR38032F, novel 5-HT3-receptor antagonist on gastric emptying in the guinea-pig

1 reference

https://api.crossref.org/works/10.1007/BF00170878

21 January 2018

Peristalsis evoked by 5-HT and renzapride: evidence for putative 5-HT4 receptor activation

1 reference

https://api.crossref.org/works/10.1007/BF00170878

21 January 2018

The gastrointestinal prokinetic benzamide derivatives are agonists at the non-classical 5-HT receptor (5-HT4) positively coupled to adenylate cyclase in neurons

1 reference

https://api.crossref.org/works/10.1007/BF00170878

21 January 2018

Azabicycloalkyl benzimidazolone derivatives as a novel class of potent agonists at the 5-HT4 receptor positively coupled to adenylate cyclase in braina

1 reference

https://api.crossref.org/works/10.1007/BF00170878

21 January 2018

Characterization of a novel 5-HT4 receptor antagonist of the azabicycloalkyl benzimidazolone class: DAU 6285

1 reference

https://api.crossref.org/works/10.1007/BF00170878

21 January 2018

Characterization of 5-HT3 and 'atypical' 5-HT receptors mediating guinea-pig ileal contractions in vitro

1 reference

https://api.crossref.org/works/10.1007/BF00170878

21 January 2018

Identification of putative 5-HT4 receptors in guinea-pig ascending colon

1 reference

https://api.crossref.org/works/10.1007/BF00170878

21 January 2018

Development of a radioligand binding assay for 5-HT4 receptors in guinea-pig and rat brain

1 reference

https://api.crossref.org/works/10.1007/BF00170878

21 January 2018

Metoclopramide. An updated review of its pharmacological properties and clinical use.

1 reference

https://api.crossref.org/works/10.1007/BF00170878

21 January 2018

The effects of metoclopramide on acetylcholine release and on smooth muscle response in the isolated guinea-pig ileum.

1 reference

https://api.crossref.org/works/10.1007/BF00170878

21 January 2018

Antiemetic activity of the new 5-HT3 antagonist DAU 6215 in animal models of cancer chemotherapy and radiation

1 reference

https://api.crossref.org/works/10.1007/BF00170878

21 January 2018

Increased gut cholinergic activity and antagonism of 5-hydroxytryptamine M-receptors by BRL 24924: potential clinical importance of BRL 24924.

1 reference

https://api.crossref.org/works/10.1007/BF00170878

21 January 2018

DAU 6285: a novel antagonist at the putative 5-HT4 receptor

1 reference

https://api.crossref.org/works/10.1007/BF00170878

21 January 2018

Novel enteric 5-HT4 receptors and gastrointestinal prokinetic action

1 reference

https://api.crossref.org/works/10.1007/BF00170878

21 January 2018

Synthesis of a new class of 2,3-dihydro-2-oxo-1H-benzimidazole-1-carboxylic acid derivatives as highly potent 5-HT3 receptor antagonists

1 reference

https://api.crossref.org/works/10.1007/BF00170878

21 January 2018

Pharmacological properties of a novel class of 5-HT3 receptor antagonists

1 reference

https://api.crossref.org/works/10.1007/BF00170878

21 January 2018

Further characterization, by use of tryptamine and benzamide derivatives, of the putative 5-HT4 receptor mediating tachycardia in the pig

1 reference

https://api.crossref.org/works/10.1007/BF00170878

21 January 2018

Identification of serotonin 5-HT3 recognition sites by radioligand binding in NG108-15 neuroblastoma-glioma cells

1 reference

https://pubmed.ncbi.nlm.nih.gov/8058105

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Relationship of serotonin-3 receptor antagonist activity to gastric emptying and motor-stimulating actions of prokinetic drugs in dogs

1 reference

https://pubmed.ncbi.nlm.nih.gov/8058105

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

AS-4370, a new gastrokinetic agent, enhances upper gastrointestinal motor activity in conscious dogs

1 reference

https://pubmed.ncbi.nlm.nih.gov/8058105

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Effects of 5-hydroxytryptamine 3 receptor antagonists on gastrointestinal motor activity in conscious dogs

1 reference

https://pubmed.ncbi.nlm.nih.gov/8058105

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Pharmacological characterization of a neuronal receptor for 5-hydroxytryptamine in guinea pig ileum with properties similar to the 5-hydroxytryptamine receptor.

1 reference

https://pubmed.ncbi.nlm.nih.gov/8058105

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The gastrointestinal motor effect of benzamide derivatives is unrelated to 5-HT3 receptor blockade

1 reference

https://pubmed.ncbi.nlm.nih.gov/8058105

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

5-Hydroxytryptamine receptor antagonism by metoclopramide and ICS 205-930 in the guinea-pig leads to enhancement of contractions of stomach muscle strips induced by electrical field stimulation and facilitation of gastric emptying in-vivo

1 reference

https://pubmed.ncbi.nlm.nih.gov/8058105

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Involvement of 5-hydroxytryptamine 3 receptors in regulation of interdigestive gastric contractions by motilin in the dog.

1 reference

https://pubmed.ncbi.nlm.nih.gov/8058105

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Hormonal control of interdigestive motor cycles of canine proximal stomach

1 reference

https://pubmed.ncbi.nlm.nih.gov/8058105

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

SC-49518 enhances gastric emptying of solid and liquid meals and stimulates gastrointestinal motility in dogs by a 5-hydroxytryptamine4 receptor mechanism.

1 reference

https://pubmed.ncbi.nlm.nih.gov/8058105

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

The novel 5-HT4 receptor antagonist DAU 6285 antagonizes 5-hydroxytryptamine-induced tachycardia in pigs

1 reference

https://pubmed.ncbi.nlm.nih.gov/8058105

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Inhibition of gastric emptying is a physiological action of cholecystokinin

1 reference

https://pubmed.ncbi.nlm.nih.gov/8058105

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Motor-stimulating properties of cisapride on isolated gastrointestinal preparations of the guinea pig.

1 reference

https://pubmed.ncbi.nlm.nih.gov/8058105

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

5-Hydroxytryptamine4 receptors mediate relaxation of the rat oesophageal tunica muscularis mucosae

1 reference

https://pubmed.ncbi.nlm.nih.gov/8058105

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Cisapride and 5-hydroxytryptamine enhance motility in the canine antrum via separate pathways, not involving 5-hydroxytryptamine1,2,3,4 receptors.

1 reference

https://pubmed.ncbi.nlm.nih.gov/8058105

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Benzimidazolone derivatives: a new class of 5-hydroxytryptamine4 receptor agonists with prokinetic and acetylcholine releasing properties in the guinea pig ileum

1 reference

https://pubmed.ncbi.nlm.nih.gov/8058105

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Effect of Proximal Gastric, Complete Gastric, and Truncal Vagotomy on Canine Gastric Electric Activity, Motility, and Emptying

1 reference

https://pubmed.ncbi.nlm.nih.gov/8058105

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Effects of cisapride on cholinergic neurotransmission and propulsive motility in the guinea pig ileum

1 reference

https://pubmed.ncbi.nlm.nih.gov/8058105

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1007/BF00170878

1 reference

Europe PubMed Central

PubMed publication ID

9 February 2018

http://europepmc.org/abstract/MED/8058105

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

9 February 2018

http://europepmc.org/abstract/MED/8058105

Sitelinks

Wikipedia(0 entries)

Wikibooks(0 entries)

Wikinews(0 entries)

Wikiquote(0 entries)

Wikisource(0 entries)

Wikiversity(0 entries)

Wikivoyage(0 entries)

Wiktionary(0 entries)

Multilingual sites(0 entries)

Retrieved from "https://www.wikidata.org/w/index.php?title=Q48146857&oldid=2209163009"