D4 dopamine receptor high-resolution structures enable the discovery of selective agonists. (Q46445025)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:29051383 AND SRC:MED&resulttype=core&format=json

7 April 2020

title

D4 dopamine receptor high-resolution structures enable the discovery of selective agonists (English)

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7 April 2020

1

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7 April 2020

Daniel Wacker

2

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7 April 2020

Anat Levit

3

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7 April 2020

Robin M Betz

5

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7 April 2020

Ron Ofer Dror

9

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7 April 2020

Brian K. Shoichet

10

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7 April 2020

Bryan L. Roth

11

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7 April 2020

author name string

Tao Che

4

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7 April 2020

John D McCorvy

6

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7 April 2020

A J Venkatakrishnan

7

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7 April 2020

Xi-Ping Huang

8

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7 April 2020

language of work or name

English

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publication date

1 October 2017

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7 April 2020

number of pages

6

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based on heuristic

inferred from page(s)

published in

Science

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volume

358

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7 April 2020

issue

6361

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7 April 2020

page(s)

381-386

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ZINC 15--Ligand Discovery for Everyone

7 April 2020

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14 June 2018

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Nonconserved residues in the second transmembrane-spanning domain of the D(4) dopamine receptor are molecular determinants of D(4)-selective pharmacology

14 June 2018

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16 June 2018

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Discovery of β-Arrestin–Biased Dopamine D 2 Ligands for Probing Signal Transduction Pathways Essential for Antipsychotic Efficacy

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PubMed

https://pubmed.ncbi.nlm.nih.gov/29051383

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Dopamine D4/D2 receptor selectivity is determined by A divergent aromatic microdomain contained within the second, third, and seventh membrane-spanning segments

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/29051383

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1126/SCIENCE.AAN5468

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:29051383 AND SRC:MED&resulttype=core&format=json

7 April 2020

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7 April 2020

PubMed publication ID

29051383

1 reference