Aromatic farnesyl diphosphate analogues: vinyl triflate-mediated synthesis and preliminary enzymatic evaluation (Q43981495)

28 November 2017

title

Aromatic farnesyl diphosphate analogues: vinyl triflate-mediated synthesis and preliminary enzymatic evaluation (English)

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28 November 2017

3

Richard A Gibbs

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28 November 2017

Chunmei Zhou

1

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28 November 2017

Ying Shao

series ordinal

2

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28 November 2017

language of work or name

English

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publication date

1 May 2002

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28 November 2017

number of pages

4

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Bioorganic & Medicinal Chemistry Letters

inferred from page(s)

published in

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28 November 2017

volume

12

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28 November 2017

issue

10

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28 November 2017

page(s)

1417-1420

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Non-peptidic prenyltransferase inhibitors: diverse structural classes and surprising anti-cancer mechanisms

28 November 2017

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Cuprate-Mediated Synthesis and Biological Evaluation of Cyclopropyl- and tert-Butylfarnesyl Diphosphate Analogs

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Grignard-mediated synthesis and preliminary biological evaluation of novel 3-substituted farnesyl diphosphate analogues

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Stereospecific synthesis and biological evaluation of farnesyl diphosphate isomers

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Synthesis and evaluation of GGPP geometric isomers: divergent substrate specificities of FTase and GGTase I.

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Crystal structure of protein farnesyltransferase at 2.25 angstrom resolution

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Cocrystal structure of protein farnesyltransferase complexed with a farnesyl diphosphate substrate

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The basis for K-Ras4B binding specificity to protein farnesyltransferase revealed by 2 A resolution ternary complex structures

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The crystal structure of human protein farnesyltransferase reveals the basis for inhibition by CaaX tetrapeptides and their mimetics

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Protein farnesyltransferase: structure and implications for substrate binding

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Crystal structure of farnesyl protein transferase complexed with a CaaX peptide and farnesyl diphosphate analogue

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Tricyclic farnesyl protein transferase inhibitors: crystallographic and calorimetric studies of structure-activity relationships

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Design and synthesis of a transferable farnesyl pyrophosphate analogue to Ras by protein farnesyltransferase

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Protein farnesyltransferase isoprenoid substrate discrimination is dependent on isoprene double bonds and branched methyl groups

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Synthesis of farnesyl diphosphate analogues containing ether-linked photoactive benzophenones and their application in studies of protein prenyltransferases

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Synthesis of Farnesol Analogues through Cu(I)-Mediated Displacements of Allylic THP Ethers by Grignard Reagents

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4 Continuous fluorescence assay for protein prenyltransferases

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Protein prenyltransferases

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Evidence for a catalytic role of zinc in protein farnesyltransferase. Spectroscopy of Co2 -farnesyltransferase indicates metal coordination of the substrate thiolate

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7 January 2021

Stereochemistry‐dependent inhibition of RAS farnesylation by farnesyl phosphonic acids

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Novel limonene phosphonate and farnesyl diphosphate analogues: design, synthesis, and evaluation as potential protein-farnesyl transferase inhibitors

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7 January 2021

10.1016/S0960-894X(02)00187-7

Identifiers

DOI

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28 November 2017

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