First "hybrid" ligands of vanilloid TRPV1 and cannabinoid CB2 receptors and non-polyunsaturated fatty acid-derived CB2-selective ligands (Q40331568)

19 September 2017

title

First "hybrid" ligands of vanilloid TRPV1 and cannabinoid CB2 receptors and non-polyunsaturated fatty acid-derived CB2-selective ligands (English)

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19 September 2017

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10

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19 September 2017

Adèle Thomas

6

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Alberto Minassi

Alberto Minassi

5

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Roger Pertwee

Roger Pertwee

8

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Giovanni Appendino

Giovanni Appendino

1

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Luciano De Petrocellis

9

Luciano De Petrocellis

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19 September 2017

Maria Grazia Cascio

2

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19 September 2017

Sara Bacchiega

3

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19 September 2017

Aniello Schiano Moriello

4

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19 September 2017

Ruth Ross

7

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19 September 2017

language of work or name

English

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publication date

29 December 2005

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19 September 2017

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19 September 2017

volume

580

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19 September 2017

issue

2

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19 September 2017

page(s)

568-574

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A comprehensive review of clinical trials on the efficacy and safety of drugs for the treatment of low back pain

19 September 2017

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Cannabinoids: a real prospect for pain relief?

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Mice lacking fatty acid amide hydrolase exhibit a cannabinoid receptor-mediated phenotypic hypoalgesia

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Reversible inhibitors of fatty acid amide hydrolase that promote analgesia: evidence for an unprecedented combination of potency and selectivity

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Overlap between the ligand recognition properties of the anandamide transporter and the VR1 vanilloid receptor: inhibitors of anandamide uptake with negligible capsaicin-like activity

21 January 2018

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Arvanil-induced inhibition of spasticity and persistent pain: evidence for therapeutic sites of action different from the vanilloid VR1 receptor and cannabinoid CB(1)/CB(2) receptors

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Highly selective CB(1) cannabinoid receptor ligands and novel CB(1)/VR(1) vanilloid receptor "hybrid" ligands

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Evidence that the plant cannabinoid Delta9-tetrahydrocannabivarin is a cannabinoid CB1 and CB2 receptor antagonist

21 January 2018

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21 January 2018

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21 January 2018

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Evidence for the involvement of the cannabinoid CB2 receptor and its endogenous ligand 2-arachidonoylglycerol in 12-O-tetradecanoylphorbol-13-acetate-induced acute inflammation in mouse ear.

21 January 2018

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2-arachidonoylglycerol, an endogenous cannabinoid receptor ligand, induces the migration of EoL-1 human eosinophilic leukemia cells and human peripheral blood eosinophils

21 January 2018

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The peripheral cannabinoid receptor Cb2, frequently expressed on AML blasts, either induces a neutrophilic differentiation block or confers abnormal migration properties in a ligand-dependent manner

21 January 2018

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21 January 2018

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10.1016/J.FEBSLET.2005.12.069

21 January 2018

Identifiers

DOI

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19 September 2017

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