Ring size in octreotide amide modulates differently agonist versus antagonist binding affinity and selectivity (Q39992321)

16 September 2017

Ring size in octreotide amide modulates differently agonist versus antagonist binding affinity and selectivity (English)

1 reference

16 September 2017

7

Jean Claude Reubi

1 reference

16 September 2017

Christy Rani R Grace

1

1 reference

16 September 2017

Judit Erchegyi

2

1 reference

16 September 2017

Manoj Samant

3

1 reference

16 September 2017

Renzo Cescato

4

1 reference

16 September 2017

Veronique Piccand

5

1 reference

16 September 2017

Roland Riek

6

1 reference

16 September 2017

Jean E Rivier

8

1 reference

16 September 2017

language of work or name

English

0 references

publication date

12 April 2008

1 reference

Journal of Medicinal Chemistry

16 September 2017

1 reference

16 September 2017

51

1 reference

16 September 2017

9

1 reference

16 September 2017

2676-2681

1 reference

Internalization of sst2, sst3, and sst5 receptors: effects of somatostatin agonists and antagonists.

16 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2789646

Torsion angle dynamics for NMR structure calculation with the new program Dyana

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2789646

Multiconformational NMR analysis of sandostatin (octreotide): equilibrium between beta-sheet and partially helical structures

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2789646

MOLMOL: a program for display and analysis of macromolecular structures

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2789646

Improved spectral resolution in cosy 1H NMR spectra of proteins via double quantum filtering

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2789646

Efficient analysis of protein 2D NMR spectra using the software packageEASY

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2789646

Peptide chemistry: development of high performance liquid chromatography and capillary zone electrophoresis

22 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2789646

Ring size of somatostatin analogues (ODT-8) modulates receptor selectivity and binding affinity

25 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2789646

Novel sst2-selective somatostatin agonists. Three-dimensional consensus structure by NMR

17 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2789646

Analysis of synthetic peptides by capillary zone electrophoresis in organic/aqueous buffers.

17 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2789646

A Refined Model for the Somatostatin Pharmacophore: Conformational Analysis of Lanthionine−Sandostatin Analogs

17 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2789646

Lanthionine-somatostatin analogs: synthesis, characterization, biological activity, and enzymatic stability studies.

17 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2789646

Three-dimensional consensus structure of sst2-selective somatostatin (SRIF) antagonists by NMR.

17 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2789646

Somatostatin receptor 1 selective analogues: 2. N(alpha)-Methylated scan

20 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2789646

Highly potent cyclic disulfide antagonists of somatostatin

20 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2789646

A selective analog for the somatostatin sst1-receptor subtype expressed by human tumors

20 August 2018

1 reference

12 December 2020

Dynamics and conformational energetics of a peptide hormone: vasopressin

1 reference

12 December 2020

Identification and characterization of novel somatostatin antagonists

1 reference

12 December 2020

Affinity profiles for human somatostatin receptor subtypes SST1-SST5 of somatostatin radiotracers selected for scintigraphic and radiotherapeutic use

1 reference

12 December 2020

Norcystine, a new tool for the study of the structure-activity relationship of peptides

1 reference

12 December 2020

Identifiers

DOI

10.1021/JM701445Q

1 reference

16 September 2017

1 reference

16 September 2017

PubMed publication ID

18410083

1 reference