Synthesis, molecular docking and biological evaluation as HDAC inhibitors of cyclopeptide mimetics by a tandem three-component reaction and intramolecular [3 2] cycloaddition. (Q39846240)

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English	Synthesis, molecular docking and biological evaluation as HDAC inhibitors of cyclopeptide mimetics by a tandem three-component reaction and intramolecular [3 2] cycloaddition.	scientific article

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29 January 2020

Synthesis, molecular docking and biological evaluation as HDAC inhibitors of cyclopeptide mimetics by a tandem three-component reaction and intramolecular [3 2] cycloaddition (English)

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29 January 2020

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Armando A. Genazzani

7

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29 January 2020

Giuseppe Bifulco

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29 January 2020

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Tracey Pirali

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29 January 2020

Valeria Faccio

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29 January 2020

Riccardo Mossetti

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29 January 2020

Ambra A Grolla

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29 January 2020

Simone Di Micco

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29 January 2020

Gian Cesare Tron

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29 January 2020

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28 May 2009

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29 January 2020

Molecular Diversity

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29 January 2020

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29 January 2020

1

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29 January 2020

109-121

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29 January 2020

Structural snapshots of human HDAC8 provide insights into the class I histone deacetylases

1 reference

https://pubmed.ncbi.nlm.nih.gov/19475493

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Homology modeling, force field design, and free energy simulation studies to optimize the activities of histone deacetylase inhibitors

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One-pot synthesis of macrocycles by a tandem three-component reaction and intramolecular [3 2] cycloaddition

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A chemical switch for the modulation of the functional activity of higher homologues of histamine on the human histamine H3 receptor: effect of various substitutions at the primary amino function

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Molecular modeling studies toward the structural optimization of new cyclopeptide-based HDAC inhibitors modeled on the natural product FR235222.

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