Synthesis and Evaluation of Quinazolone Derivatives as a New Class of c-KIT G-Quadruplex Binding Ligands. (Q38988080)

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20 March 2020

title

Synthesis and Evaluation of Quinazolone Derivatives as a New Class of c-KIT G-Quadruplex Binding Ligands (English)

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3

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author name string

Xiaoxiao Wang

1

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20 March 2020

Chen-Xi Zhou

2

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20 March 2020

Jin-Qiang Hou

4

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20 March 2020

Shuo-Bin Chen

5

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20 March 2020

Tian-Miao Ou

6

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20 March 2020

Lian-Quan Gu

7

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Zhi-Shu Huang

8

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20 March 2020

Jia-Heng Tan

9

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20 March 2020

publication date

13 August 2013

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ACS Medicinal Chemistry Letters

20 March 2020

published in

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volume

4

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issue

10

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page(s)

909-914

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Crystal structure of a c-kit promoter quadruplex reveals the structural role of metal ions and water molecules in maintaining loop conformation

20 March 2020

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Facilitation of a structural transition in the polypurine/polypyrimidine tract within the proximal promoter region of the human VEGF gene by the presence of potassium and G-quadruplex-interactive agents

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21 August 2018

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Folate analogues. 35. Synthesis and biological evaluation of 1-deaza, 3-deaza, and bridge-elongated analogues of N10-propargyl-5,8-dideazafolic acid

21 August 2018

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PubMed

https://pubmed.ncbi.nlm.nih.gov/24900584

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1021/ML400271Y

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20 March 2020

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20 March 2020

PubMed publication ID

24900584

1 reference

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