Refining stability and dissolution rate of amorphous drug formulations (Q38206296)

31 August 2017

title

Refining stability and dissolution rate of amorphous drug formulations (English)

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31 August 2017

8

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31 August 2017

Petra Alexandra Priemel

Petra A Priemel

2

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Line Hagner Nielsen

Line Hagner Nielsen

4

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Korbinian Löbmann

Korbinian Löbmann

3

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Holger Grohganz

Holger Grohganz

1

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Riikka Laitinen

5

Riikka Laitinen

1 reference

31 August 2017

Anette Mullertz

6

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31 August 2017

Guy Van den Mooter

7

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31 August 2017

language of work or name

English

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publication date

23 April 2014

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Expert Opinion on Drug Delivery

31 August 2017

published in

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31 August 2017

volume

11

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31 August 2017

issue

6

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31 August 2017

page(s)

977-989

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A theoretical basis for a biopharmaceutic drug classification: the correlation of in vitro drug product dissolution and in vivo bioavailability

31 August 2017

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Solid dispersions: a strategy for poorly aqueous soluble drugs and technology updates

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Phase behavior of amorphous molecular dispersions I: Determination of the degree and mechanism of solid solubility

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Solubilities of crystalline drugs in polymers: an improved analytical method and comparison of solubilities of indomethacin and nifedipine in PVP, PVP/VA, and PVAc

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Theoretical and practical approaches for prediction of drug-polymer miscibility and solubility.

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Influence of preparation methods on solid state supersaturation of amorphous solid dispersions: a case study with itraconazole and eudragit e100.

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A method to predict the equilibrium solubility of drugs in solid polymers near room temperature using thermal analysis

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Construction of drug-polymer thermodynamic phase diagrams using Flory-Huggins interaction theory: identifying the relevance of temperature and drug weight fraction to phase separation within solid dispersions

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Characterization of carbamazepine-Gelucire 50/13 microparticles prepared by a spray-congealing process using ultrasounds.

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Melt extrusion: from process to drug delivery technology

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Fusion processing of itraconazole solid dispersions by kinetisol dispersing: a comparative study to hot melt extrusion

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Applications of supercritical fluids to enhance the dissolution behaviors of Furosemide by generation of microparticles and solid dispersions

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Processing of carbamazepine-PEG 4000 solid dispersions with supercritical carbon dioxide: preparation, characterisation, and in vitro dissolution

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The effect of pressurized carbon dioxide as a temporary plasticizer and foaming agent on the hot stage extrusion process and extrudate properties of solid dispersions of itraconazole with PVP-VA 64.

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Spatial confinement can lead to increased stability of amorphous indomethacin

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Stability of amorphous pharmaceutical solids: crystal growth mechanisms and effect of polymer additives

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Fast surface crystallization of amorphous griseofulvin below T g.

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Surface-enhanced crystallization of amorphous nifedipine

21 January 2018

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Glasses crystallize rapidly at free surfaces by growing crystals upward

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Aqueous film coating to reduce recrystallization of guaifenesin from hot-melt extruded acrylic matrices

21 January 2018

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Stabilisation of amorphous drugs under high humidity using pharmaceutical thin films.

21 January 2018

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Phase behavior of poly(vinylpyrrolidone) containing amorphous solid dispersions in the presence of moisture.

21 January 2018

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Mesoporous systems for poorly soluble drugs

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Application of Mesoporous Silicon Dioxide and Silicate in Oral Amorphous Drug Delivery Systems

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Physical state of poorly water soluble therapeutic molecules loaded into SBA-15 ordered mesoporous silica carriers: a case study with itraconazole and ibuprofen

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Oxidized mesoporous silicon microparticles for improved oral delivery of poorly soluble drugs

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Physical characterization and stability of amorphous indomethacin and ranitidine hydrochloride binary systems prepared by mechanical activation

21 January 2018

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Enhanced dissolution rate and synchronized release of drugs in binary systems through formulation: Amorphous naproxen-cimetidine mixtures prepared by mechanical activation

21 January 2018

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Coamorphous drug systems: enhanced physical stability and dissolution rate of indomethacin and naproxen.

21 January 2018

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A theoretical and spectroscopic study of co-amorphous naproxen and indomethacin

21 January 2018

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Amino acids as co-amorphous stabilizers for poorly water soluble drugs--Part 1: preparation, stability and dissolution enhancement

21 January 2018

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Amino acids as co-amorphous stabilizers for poorly water-soluble drugs--Part 2: molecular interactions.

21 January 2018

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Amorphous pharmaceutical solids: preparation, characterization and stabilization

21 January 2018

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Improved physical stability of amorphous state through acid base interactions

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Coamorphous repaglinide-saccharin with enhanced dissolution

21 January 2018

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Studies on dissolution enhancement and mathematical modeling of drug release of a poorly water-soluble drug using water-soluble carriers

21 January 2018

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Cocrystallization and amorphization induced by drug-excipient interaction improves the physical properties of acyclovir.

21 January 2018

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Impact of process variables on the micromeritic and physicochemical properties of spray-dried porous microparticles, part I: introduction of a new morphology classification system

21 January 2018

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Effect of counterions on the properties of amorphous atorvastatin salts

21 January 2018

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Modification of the solid-state nature of sulfathiazole and sulfathiazole sodium by spray drying

21 January 2018

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Impact of process variables on the micromeritic and physicochemical properties of spray-dried microparticles--Part II. Physicochemical characterisation of spray-dried materials

21 January 2018

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Bulk, surface properties and water uptake mechanisms of salt/acid amorphous composite systems

21 January 2018

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Influence of tablet dissolution on furosemide bioavailability: a bioequivalence study.

21 January 2018

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Preparation of an amorphous sodium furosemide salt improves solubility and dissolution rate and leads to a faster Tmax after oral dosing to rats

21 January 2018

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https://api.crossref.org/works/10.1517/17425247.2014.911728

Biorelevant characterisation of amorphous furosemide salt exhibits conversion to a furosemide hydrate during dissolution

21 January 2018

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https://api.crossref.org/works/10.1517/17425247.2014.911728

In situ amorphisation of indomethacin with Eudragit® E during dissolution

21 January 2018

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https://api.crossref.org/works/10.1517/17425247.2014.911728

A comparative study of the effect of spray drying and hot-melt extrusion on the properties of amorphous solid dispersions containing felodipine.

21 January 2018

1 reference

https://api.crossref.org/works/10.1517/17425247.2014.911728

Evaluation of drug supersaturation by thermodynamic and kinetic approaches for the prediction of oral absorbability in amorphous pharmaceuticals

21 January 2018

1 reference

https://api.crossref.org/works/10.1517/17425247.2014.911728

Evaluation of the structural determinants of polymeric precipitation inhibitors using solvent shift methods and principle component analysis.

21 January 2018

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https://api.crossref.org/works/10.1517/17425247.2014.911728

Drug precipitation-permeation interplay: supersaturation in an absorptive environment

21 January 2018

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https://api.crossref.org/works/10.1517/17425247.2014.911728

Precipitation in and Supersaturation of Contents of the Upper Small Intestine After Administration of Two Weak Bases to Fasted Adults

21 January 2018

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https://api.crossref.org/works/10.1517/17425247.2014.911728

Precipitation of a poorly soluble model drug during in vitro lipolysis: characterization and dissolution of the precipitate

21 January 2018

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https://api.crossref.org/works/10.1517/17425247.2014.911728

Miniaturized screening of polymers for amorphous drug stabilization (SPADS): Rapid assessment of solid dispersion systems

21 January 2018

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https://api.crossref.org/works/10.1517/17425247.2014.911728

In vitro and in vivo performance of novel supersaturated self-nanoemulsifying drug delivery systems (super-SNEDDS)

21 January 2018

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https://api.crossref.org/works/10.1517/17425247.2014.911728

The impact of surface- and nano-crystallisation on the detected amorphous content and the dissolution behaviour of amorphous indomethacin

21 January 2018

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https://api.crossref.org/works/10.1517/17425247.2014.911728

Inhibition of surface crystallisation of amorphous indomethacin particles in physical drug–polymer mixtures

21 January 2018

1 reference

https://api.crossref.org/works/10.1517/17425247.2014.911728

Co-amorphous simvastatin and glipizide combinations show improved physical stability without evidence of intermolecular interactions

21 January 2018

1 reference

https://api.crossref.org/works/10.1517/17425247.2014.911728

Effect of different preparation methods on the dissolution behaviour of amorphous indomethacin

21 January 2018

1 reference

https://api.crossref.org/works/10.1517/17425247.2014.911728

Preparation of glass solutions of three poorly water soluble drugs by spray drying, melt extrusion and ball milling

21 January 2018

1 reference

https://api.crossref.org/works/10.1517/17425247.2014.911728

10.1517/17425247.2014.911728

21 January 2018

Identifiers

DOI

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31 August 2017

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