Recent advances in the development of melatonin MT(1) and MT(2) receptor agonists. (Q37763715)

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5 February 2020

review article

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title

Recent advances in the development of melatonin MT(1) and MT(2) receptor agonists (English)

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5 February 2020

Silvia Rivara

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5 February 2020

Daniele Pala

3

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5 February 2020

Annalida Bedini

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5 February 2020

Gilberto Spadoni

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5 February 2020

6

Giorgio Tarzia

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5 February 2020

language of work or name

English

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publication date

1 August 2010

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Expert Opinion on Therapeutic Patents

5 February 2020

published in

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5 February 2020

volume

20

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issue

8

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5 February 2020

page(s)

1059-1077

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Persistence of circadian rhythmicity in a mammalian hypothalamic "island" containing the suprachiasmatic nucleus

5 February 2020

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Melatonin as a naturally occurring co-substrate of quinone reductase-2, the putative MT3 melatonin membrane receptor: hypothesis and significance

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Reduced hippocampal MT2 melatonin receptor expression in Alzheimer's disease.

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The regional and cellular expression profile of the melatonin receptor MT1 in the central dopaminergic system

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The melatonin receptor subtype MT2 is present in the human cardiovascular system

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Distribution of melatonin MT1 receptor immunoreactivity in human retina

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Melatonin in rheumatoid arthritis: synovial macrophages show melatonin receptors

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Targeted disruption of the mouse Mel(1b) melatonin receptor

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Rhythmic gene expression in pituitary depends on heterologous sensitization by the neurohormone melatonin

21 January 2018

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Melatonin receptor antagonists that differentiate between the human Mel1a and Mel1b recombinant subtypes are used to assess the pharmacological profile of the rabbit retina ML1 presynaptic heteroreceptor

21 January 2018

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Constitutively active melatonin MT(1) receptors in male rat caudal arteries

21 January 2018

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MT(2) melatonin receptors are present and functional in rat caudal artery

21 January 2018

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Melatonin and melatonergic drugs on sleep: possible mechanisms of action

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Circadian misalignment in mood disturbances

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The pattern of melatonin receptor expression in the brain may influence antidepressant treatment

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Antiepileptic activity of melatonin in guinea pigs with pentylenetetrazol-induced seizures

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Effects of melatonin in experimental stroke models in acute, sub-acute, and chronic stages

21 January 2018

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Melatonin inhibits estrogen receptor transactivation and cAMP levels in breast cancer cells

21 January 2018

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Investigational melatonin receptor agonists

21 January 2018

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Melatonin agonist tasimelteon (VEC-162) for transient insomnia after sleep-time shift: two randomised controlled multicentre trials.

21 January 2018

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Melatonin receptor agonists: SAR and applications to the treatment of sleep-wake disorders

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Recent advances in melatonin receptor ligands.

21 January 2018

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Binding affinity and biological activity of oxygen and sulfur isosteres at melatonin receptors as a function of their hydrogen bonding capability

21 January 2018

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Bicyclic melatonin receptor agonists containing a ring-junction nitrogen: Synthesis, biological evaluation, and molecular modeling of the putative bioactive conformation

21 January 2018

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Synthesis of new tricyclic melatoninergic ligands

21 January 2018

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Synthesis and biological evaluation of new β,β′-disubstituted 6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl ethylamido melatoninergic ligands

21 January 2018

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Conformationally restrained melatonin analogues: synthesis, binding affinity for the melatonin receptor, evaluation of the biological activity, and molecular modeling study

21 January 2018

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Reassessing the melatonin pharmacophore--enantiomeric resolution, pharmacological activity, structure analysis, and molecular modeling of a constrained chiral melatonin analogue

21 January 2018

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Mapping the melatonin receptor. 6. Melatonin agonists and antagonists derived from 6H-isoindolo[2,1-a]indoles, 5,6-dihydroindolo[2,1-a]isoquinolines, and 6,7-dihydro-5H-benzo[c]azepino[2,1-a]indoles

21 January 2018

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Sleep-promoting action of IIK7, a selective MT2 melatonin receptor agonist in the rat

21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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N-(substituted-anilinoethyl)amides: design, synthesis, and pharmacological characterization of a new class of melatonin receptor ligands

21 January 2018

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Synthesis of substituted N-[3-(3-methoxyphenyl)propyl] amides as highly potent MT(2)-selective melatonin ligands.

21 January 2018

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Melatonin and enterochromaffine cells

21 January 2018

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The Efficacy and Safety of the Melatonin Agonist beta-Methyl-6-Chloromelatonin in Primary Insomnia

21 January 2018

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10.1517/13543776.2010.496455

21 January 2018

Identifiers

DOI

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20533893 AND SRC:MED&resulttype=core&format=json

5 February 2020

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