Acyl hydroxypyrazoles as novel agonists for high-affinity nicotinic acid receptor GPR109A: WO2008051403. (Q37536057)

20 August 2017

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title

Acyl hydroxypyrazoles as novel agonists for high-affinity nicotinic acid receptor GPR109A: WO2008051403. (English)

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20 August 2017

Hong C Shen

1

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20 August 2017

language of work or name

English

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publication date

1 August 2009

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Expert Opinion on Therapeutic Patents

20 August 2017

published in

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20 August 2017

volume

19

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20 August 2017

issue

8

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20 August 2017

page(s)

1149-1155

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One-year reduction and longitudinal analysis of carotid intima-media thickness associated with colestipol/niacin therapy

20 August 2017

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PUMA-G and HM74 are receptors for nicotinic acid and mediate its anti-lipolytic effect

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Discovery of biaryl anthranilides as full agonists for the high affinity niacin receptor

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3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydro-cyclopentapyrazole (MK-0354): a partial agonist of the nicotinic acid receptor, G-protein coupled receptor 109a, with antilipolytic but no vasodilatory activity in mice.

21 January 2018

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Effects of a niacin receptor partial agonist, MK-0354, on plasma free fatty acids, lipids, and cutaneous flushing in humans

21 January 2018

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Nicotinic acid receptor agonists

21 January 2018

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Characterization of determinants of ligand binding to the nicotinic acid receptor GPR109A (HM74A/PUMA-G).

21 January 2018

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Molecular modeling aided design of nicotinic acid receptor GPR109A agonists

21 January 2018

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Tetrahydro anthranilic acid as a surrogate for anthranilic acid: application to the discovery of potent niacin receptor agonists

21 January 2018

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Identifiers

DOI

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20 August 2017

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