Systemic administration of the adenosine A(2A) agonist CGS 21680 induces sedation at doses that suppress lever pressing and food intake (Q37172329)

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2 January 2020

title

Systemic administration of the adenosine A(2A) agonist CGS 21680 induces sedation at doses that suppress lever pressing and food intake (English)

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2 January 2020

4

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2 January 2020

John D. Salamone

5

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2 January 2020

author name string

Susana Mingote

1

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2 January 2020

Mariana Pereira

2

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2 January 2020

Andrew M Farrar

3

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2 January 2020

language of work or name

English

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publication date

17 January 2008

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Pharmacology, Biochemistry and Behavior

2 January 2020

published in

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2 January 2020

volume

89

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2 January 2020

issue

3

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2 January 2020

page(s)

345-351

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Potential role of adenosine A2A receptors in the treatment of schizophrenia

2 January 2020

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The adenosine A2A receptor agonist, CGS-21680, blocks excessive rearing, acquisition of wheel running, and increases nucleus accumbens CREB phosphorylation in chronically food-restricted rats.

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Scopolamine reverses haloperidol-attenuated lever-pressing for water but not haloperidol-attenuated water intake in the rat

6 September 2017

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Injections of the selective adenosine A2A antagonist MSX-3 into the nucleus accumbens core attenuate the locomotor suppression induced by haloperidol in rats.

28 September 2017

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The adenosine A2A receptor agonist CGS 21680 exhibits antipsychotic-like activity in Cebus apella monkeys

27 June 2018

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An adenosine A2a agonist increases sleep and induces Fos in ventrolateral preoptic neurons.

27 June 2018

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27 June 2018

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Different behavioral effects of haloperidol, clozapine and thioridazine in a concurrent lever pressing and feeding procedure.

27 June 2018

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The role of brain dopamine in response initiation: effects of haloperidol and regionally specific dopamine depletions on the local rate of instrumental responding.

27 June 2018

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27 June 2018

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3 September 2018

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3 September 2018

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3 September 2018

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The cannabinoid CB1 antagonist AM 251 produces food avoidance and behaviors associated with nausea but does not impair feeding efficiency in rats.

3 September 2018

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An adenosine A receptor agonist induces sleep by increasing GABA release in the tuberomammillary nucleus to inhibit histaminergic systems in rats.

3 September 2018

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The adenosine A2A antagonist KF17837 reverses the locomotor suppression and tremulous jaw movements induced by haloperidol in rats: possible relevance to parkinsonism.

3 September 2018

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Behavioral effects of inhibition of cannabinoid metabolism: The amidase inhibitor AM374 enhances the suppression of lever pressing produced by exogenously administered anandamide

3 September 2018

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Involvement of adenosine A1 and A2A receptors in the adenosinergic modulation of the discriminative-stimulus effects of cocaine and methamphetamine in rats

3 September 2018

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Influence of CGS 21680, a selective adenosine A(2A) agonist, on the phencyclidine-induced sensorimotor gating deficit and motor behaviour in rats

3 September 2018

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3 September 2018

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Dopamine antagonists alter response allocation but do not suppress appetite for food in rats: contrast between the effects of SKF 83566, raclopride, and fenfluramine on a concurrent choice task

3 September 2018

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3 September 2018

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Catalepsy induced by a blockade of dopamine D1 or D2 receptors was reversed by a concomitant blockade of adenosine A(2A) receptors in the caudate-putamen of rats

3 September 2018

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3 September 2018

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SCH 58261, an A(2A) adenosine receptor antagonist, counteracts parkinsonian-like muscle rigidity in rats

3 September 2018

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Caffeine and schizophrenia.

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3 September 2018

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Motor depressant effects mediated by dopamine D2 and adenosine A2A receptors in the nucleus accumbens and the caudate-putamen

3 September 2018

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Adenosine A2a receptors in the nucleus accumbens mediate locomotor depression

3 September 2018

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Ventrolateral striatal dopamine depletions impair feeding and food handling in rats

3 September 2018

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Direct autoradiographic localization of adenosine A2 receptors in the rat brain using the A2-selective agonist, [3H]CGS 21680

3 September 2018

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12 December 2020

Adenosine/dopamine interaction: implications for the treatment of Parkinson's disease

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Effects of acute and repeated clozapine injections on cholinomimetic-induced vacuous jaw movements

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Characterisation of adjustments to the structure of feeding behaviour following pharmacological treatment: effects of amphetamine and fenfluramine and the antagonism produced by pimozide and methergoline

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Caffeine: use and effects in long-stay psychiatric patients

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Effects of caffeine in chronic psychiatric patients

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10.1016/J.PBB.2008.01.006

Identifiers

DOI

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:18281083 AND SRC:MED&resulttype=core&format=json

2 January 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:18281083 AND SRC:MED&resulttype=core&format=json

2 January 2020

PubMed publication ID

18281083

1 reference