Estrogen receptor (ER) modulators each induce distinct conformational changes in ER alpha and ER beta. (Q36456030)

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12 November 2019

title

Estrogen receptor (ER) modulators each induce distinct conformational changes in ER alpha and ER beta (English)

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12 November 2019

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9

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12 November 2019

author name string

L A Paige

1

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12 November 2019

D J Christensen

2

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H Grøn

3

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J D Norris

4

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E B Gottlin

5

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K M Padilla

6

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C Y Chang

7

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L M Ballas

8

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D P McDonnell

10

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D M Fowlkes

11

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12 November 2019

language of work or name

English

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publication date

1 March 1999

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Proceedings of the National Academy of Sciences of the United States of America

12 November 2019

published in

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volume

96

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issue

7

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12 November 2019

page(s)

3999-4004

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The structural basis of estrogen receptor/coactivator recognition and the antagonism of this interaction by tamoxifen

12 November 2019

cites work

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=22409

Estrogen receptor alpha requires no accessory factors for high-affinity binding to a consensus response element

30 September 2017

1 reference

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Basic guide to the mechanisms of antiestrogen action

30 September 2017

1 reference

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Enhancement of estrogen receptor transcriptional activity by the coactivator GRIP-1 highlights the role of activation function 2 in determining estrogen receptor pharmacology

30 September 2017

1 reference

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Diverse signaling pathways modulate nuclear receptor recruitment of N-CoR and SMRT complexes

30 September 2017

1 reference

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Functional role of estrogen metabolism in target cells: review and perspectives

30 September 2017

1 reference

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Pharmacokinetics and Pharmacodynamics of Conjugated Equine Estrogens: Chemistry and Metabolism

30 September 2017

1 reference

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Molecular determinants of tissue selectivity in estrogen receptor modulators

30 September 2017

1 reference

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Molecular basis of agonism and antagonism in the oestrogen receptor

30 September 2017

1 reference

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A signature motif in transcriptional co-activators mediates binding to nuclear receptors

30 September 2017

1 reference

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Antiestrogens: future prospects.

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=22409

ER beta: identification and characterization of a novel human estrogen receptor

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=22409

Cloning of a novel receptor expressed in rat prostate and ovary

30 September 2017

1 reference

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Steroid receptors and their associated proteins

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=22409

Raloxifene (LY139481 HCI) prevents bone loss and reduces serum cholesterol without causing uterine hypertrophy in ovariectomized rats

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=22409

Sequence and characterization of a coactivator for the steroid hormone receptor superfamily

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=22409

Sequence and expression of human estrogen receptor complementary DNA

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=22409

Zinc fingers: gilt by association

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=22409

In situ distinction between steroid receptor binding and transactivation at a target gene

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=22409

The strategic use of antiestrogens to control the development and growth of breast cancer.

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=22409

Effects of tamoxifen on bone mineral density in postmenopausal women with breast cancer

30 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=22409

Analysis of estrogen receptor function in vitro reveals three distinct classes of antiestrogens

30 September 2017

1 reference

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Mechanisms of Cardioprotection by Estrogens

30 September 2017

1 reference

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Coactivator and corepressor regulation of the agonist/antagonist activity of the mixed antiestrogen, 4-hydroxytamoxifen.

28 June 2018

1 reference

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William L. McGuire Memorial Lecture. Antiestrogens: mechanisms of action and resistance in breast cancer

28 June 2018

1 reference

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Transcriptional activation by the estrogen receptor requires a conformational change in the ligand binding domain

28 June 2018

1 reference

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Pharmacokinetics of 17 beta-dihydroequilin sulfate and 17 beta-dihydroequilin in normal postmenopausal women

28 June 2018

1 reference

12 December 2020

Effects of tamoxifen on uterus and ovaries of postmenopausal women in a randomised breast cancer prevention trial

1 reference

12 December 2020

Effect of 17α-Dihydroequilin Sulfate, a Conjugated Equine Estrogen, and Ethynylestradiol on Atherosclerosis in Cholesterol-Fed Rabbits

1 reference

12 December 2020

Synthesis and pharmacology of conformationally restricted raloxifene analogues: highly potent selective estrogen receptor modulators

1 reference

12 December 2020

Identifiers

DOI

10.1073/PNAS.96.7.3999

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:10097152 AND SRC:MED&resulttype=core&format=json

12 November 2019

0 references

1 reference

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12 November 2019

PubMed publication ID

10097152

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