SST3-selective potent peptidic somatostatin receptor antagonists (Q35582980)

9 August 2017

title

SST3-selective potent peptidic somatostatin receptor antagonists (English)

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9 August 2017

J C Reubi

1

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9 August 2017

J C Schaer

2

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9 August 2017

S Wenger

3

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9 August 2017

C Hoeger

4

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9 August 2017

J Erchegyi

5

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9 August 2017

B Waser

6

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9 August 2017

J Rivier

7

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9 August 2017

language of work or name

English

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publication date

1 December 2000

1 reference

Proceedings of the National Academy of Sciences of the United States of America

9 August 2017

published in

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9 August 2017

volume

97

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9 August 2017

issue

25

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9 August 2017

page(s)

13973-13978

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(R)-tert-Butoxycarbonylamino-fluorenylmethoxycarbonyl-glycine from (S)-benzyloxycarbonyl-serine or from papain resolution of the corresponding amide or methyl ester

9 August 2017

cites work

1 reference

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12 July 2018

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Visualisation of somatostatin receptor sst(3) in the rat central nervous system

12 July 2018

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Expression of somatostatin receptor subtypes on guinea pig gastric and colonic smooth muscle cells.

12 July 2018

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Selective targeting of somatostatin receptor 3 to neuronal cilia

12 July 2018

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Rapid identification of subtype-selective agonists of the somatostatin receptor through combinatorial chemistry

12 July 2018

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Mack Forster Award Lecture Receptor nuclear medicine: vasointestinal peptide and somatostatin receptor scintigraphy for diagnosis and treatment of tumour patients

12 July 2018

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Betidamino Acid Scan of the GnRH Antagonist Acyline

12 July 2018

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ActivationIn Vitroof Somatostatin Receptor Subtypes 2, 3, or 4 Stimulates Protein Tyrosine Phosphatase Activity in Membranes from Transfected Ras-Transformed NIH 3T3 Cells: Coexpression with Catalytically Inactive SHP-2 Blocks Responsiveness

12 July 2018

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Involvement of MAP kinase and c-fos signaling in the inhibition of cell growth by somatostatin

12 July 2018

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Subtype-selective induction of wild-type p53 and apoptosis, but not cell cycle arrest, by human somatostatin receptor 3

12 July 2018

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Somatostatin receptor-mediated signaling in smooth muscle. Activation of phospholipase C-beta3 by Gbetagamma and inhibition of adenylyl cyclase by Galphai1 and Galphao

12 July 2018

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12 July 2018

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12 July 2018

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Activation of a protein tyrosine phosphatase and inactivation of Raf-1 by somatostatin

12 July 2018

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Loss of sst2 somatostatin receptor gene expression in human pancreatic and colorectal cancer.

12 July 2018

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Stimulation of tyrosine phosphatase and inhibition of cell proliferation by somatostatin analogues: mediation by human somatostatin receptor subtypes SSTR1 and SSTR2.

12 July 2018

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Inhibition of cell proliferation by the somatostatin analogue RC-160 is mediated by somatostatin receptor subtypes SSTR2 and SSTR5 through different mechanisms

12 July 2018

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Classification and nomenclature of somatostatin receptors

12 July 2018

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Somatostatin receptor subtype gene expression in pituitary adenomas

12 July 2018

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12 July 2018

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Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

12 July 2018

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Highly potent cyclic disulfide antagonists of somatostatin

12 July 2018

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Different expression patterns of somatostatin receptor subtypes in cultured epithelial cells from human normal prostate and prostate cancer

26 September 2018

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Heterogeneous expression of two somatostatin receptor subtypes in pituitary tumors

26 September 2018

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Somatostatin receptor subtype gene expression in pituitary adenomas

26 September 2018

1 reference

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High incidence of somatostatin receptors in human meningiomas: biochemical characterization

26 September 2018

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Subtype-selective induction of wild-type p53 and apoptosis, but not cell cycle arrest, by human somatostatin receptor 3

26 September 2018

1 reference

Crossref

https://api.crossref.org/works/10.1073/PNAS.250483897

Somatostatin receptor subtype 3 mediates the inhibitory action of somatostatin on gastric smooth muscle cells

21 January 2018

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12 December 2020

In vitro identification of vasoactive intestinal peptide receptors in human tumors: implications for tumor imaging

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12 December 2020

Molecular biology of somatostatin receptors

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12 December 2020

Somatostatin receptor subtypes sst1, sst2, sst3 and sst5 expression in human pituitary, gastroentero-pancreatic and mammary tumors: comparison of mRNA analysis with receptor autoradiography

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12 December 2020

Antagonist-stimulated internalization of the G protein-coupled cholecystokinin receptor

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12 December 2020

Somatostatin increases mitogen-induced IL-2 secretion and proliferation of human jurkat T cells via sst3 receptor isotype

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12 December 2020

Yttrium-90-labelled somatostatin-analogue for cancer treatment

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12 December 2020

Affinity profiles for human somatostatin receptor subtypes SST1-SST5 of somatostatin radiotracers selected for scintigraphic and radiotherapeutic use

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12 December 2020

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12 December 2020

Detection of somatostatin receptors in surgical and percutaneous needle biopsy samples of carcinoids and islet cell carcinomas

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12 December 2020

New method for the synthesis of N-methyl amino acids containing peptides by reductive methylation of amino groups on the solid phase

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12 December 2020

Expression and localization of somatostatin receptor SSTR1, SSTR2, and SSTR3 messenger RNAs in primary human tumors using in situ hybridization

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12 December 2020

Expression of Somatostatin Receptor Subtype 1–5 Genes in Human Pancreatic Cancer

1 reference

12 December 2020

Immunohistochemical detection of somatostatin sst2a receptors in the lymphatic, smooth muscular, and peripheral nervous systems of the human gastrointestinal tract: facts and artifacts

1 reference

12 December 2020

Identifiers

DOI

10.1073/PNAS.250483897

1 reference

9 August 2017

0 references

1 reference

9 August 2017

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