SB-258741: a 5-HT7 receptor antagonist of potential clinical interest. (Q34692022)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12070528 AND SRC:MED&resulttype=core&format=json

10 November 2019

review article

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title

SB-258741: a 5-HT7 receptor antagonist of potential clinical interest (English)

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12070528 AND SRC:MED&resulttype=core&format=json

10 November 2019

author name string

Bruno Pouzet

series ordinal

1

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12070528 AND SRC:MED&resulttype=core&format=json

10 November 2019

publication date

1 January 2002

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12070528 AND SRC:MED&resulttype=core&format=json

CNS Neuroscience & Therapeutics

10 November 2019

published in

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10 November 2019

volume

8

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10 November 2019

issue

1

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10 November 2019

page(s)

90-100

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Hyper- and hypoaldosteronism

10 November 2019

cites work

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Changes in systemic and regional haemodynamics during 5-HT7 receptor-mediated depressor responses in rats

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Pharmacological evidence for the 5-HT7 receptor mediating smooth muscle relaxation in canine cerebral arteries

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Central mechanisms of pain modulation

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Effects of antidepressants on 5-HT7 receptor regulation in the rat hypothalamus

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A review of central 5-HT receptors and their function

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Pharmacological and molecular characterization of 5-hydroxytryptamine(7) receptors in the rat adrenal gland

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Involvement of serotonin 2A receptors in phencyclidine-induced disruption of prepulse inhibition of the acoustic startle in rats

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5-CT stimulation of adenylyl cyclase activity in guinea-pig hippocampus: evidence for involvement of 5-HT7 and 5-HT1A receptors

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A novel, potent, and selective 5-HT(7) antagonist: (R)-3-(2-(2-(4-methylpiperidin-1-yl)ethyl)pyrrolidine-1-sulfonyl) phen ol (SB-269970).

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12 December 2020

[(3)H]-SB-269970--A selective antagonist radioligand for 5-HT(7) receptors

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12 December 2020

Characterization of SB-269970-A, a selective 5-HT(7) receptor antagonist

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12 December 2020

The treatment of bipolar depression.

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Animal models of deficient sensorimotor gating: what we know, what we think we know, and what we hope to know soon

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Effect of serotonergic drugs on footshock-induced ultrasonic vocalization in adult male rats

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Phencyclidine-induced stereotyped behaviour and social isolation in rats: a possible animal model of schizophrenia.

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12 December 2020

The effect of SB-269970, a 5-HT(7) receptor antagonist, on 5-HT release from serotonergic terminals and cell bodies

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12 December 2020

Role of 5-HT(1A) and 5-HT(7) receptors in the facilitatory response induced by 8-OH-DPAT on learning consolidation

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In vivo resetting of the hamster circadian clock by 5-HT7 receptors in the suprachiasmatic nucleus.

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Effects of acute versus chronic treatment with typical or atypical antipsychotics on d-amphetamine-induced sensorimotor gating deficits in rats

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Chronic pain, chronic stress and depression: coincidence or consequence?

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12 December 2020

Effects of the 5-HT(7) receptor antagonist SB-258741 in animal models for schizophrenia

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Phase Advance of the Circadian Sleep-Wake Cycle as an Antidepressant

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12 December 2020

Inhibition of shock-elicited ultrasonic vocalization by opioid peptides in the rat: a psychotropic effect

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Effects of phencyclidine and phencyclidine biologs on sensorimotor gating in the rat.

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Optimizing the pentetrazol infusion test for seizure threshold measurement.

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Effects of housing and muricidal behavior on serotonergic receptors and interactions with novel anxiolytic drugs

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Basal ganglia and limbic system pathology in schizophrenia. A morphometric study of brain volume and shrinkage

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Depression: a new animal model sensitive to antidepressant treatments

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Behavioral despair in mice: a primary screening test for antidepressants

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Pharmacological Specificity of Conditioned Avoidance Response Inhibition in Rats: Inhibition by Neuroleptics and Correlation to Dopamine Receptor Blockade

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[Study approach and initial results of the effect of sleep deprivation on the depressive syndrome]

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Antinociceptive and anticonvulsive effect of THIP, a pure GABA agonist

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Antipsychotic agents antagonize non-competitive N-methyl-D-aspartate antagonist-induced behaviors

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12 December 2020

Differential effects of classical and newer antipsychotics on the hypermotility induced by two dose levels of D-amphetamine

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12 December 2020

Cloning and expression of a 5-hydroxytryptamine7 receptor positively coupled to adenylyl cyclase

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Do antidepressants stabilize mood through actions on the hypothalamic-pituitary-adrenocortical system?

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12 December 2020

Characterization and distribution of putative 5-ht7 receptors in guinea-pig brain

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12 December 2020

Expression of serotonin receptor mRNAs in blood vessels

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12 December 2020

Cloning and expression of a novel serotonin receptor with high affinity for tricyclic psychotropic drugs

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12 December 2020

Identification of 5-hydroxytryptamine7 receptor binding sites in rat hypothalamus: sensitivity to chronic antidepressant treatment

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12 December 2020

Binding of typical and atypical antipsychotic agents to 5-hydroxytryptamine-6 and 5-hydroxytryptamine-7 receptors

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12 December 2020

Clozapine antagonizes phencyclidine-induced deficits in sensorimotor gating of the startle response.

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12 December 2020

Molecular cloning and expression of a 5-hydroxytryptamine7 serotonin receptor subtype

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12 December 2020

Molecular cloning, characterization, and localization of a high-affinity serotonin receptor (5-HT7) activating cAMP formation

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12 December 2020

A novel adenylyl cyclase-activating serotonin receptor (5-HT7) implicated in the regulation of mammalian circadian rhythms

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12 December 2020

A clinician's primer on the circadian clock: its localization, function, and resetting

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12 December 2020

Serotonin and the mammalian circadian system: I. In vitro phase shifts by serotonergic agonists and antagonists

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12 December 2020

Sleep research in depressive illness: clinical implications--a tasting menu

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12 December 2020

Pressure natriuresis and long-term blood pressure control.

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12 December 2020

A receptor autoradiographic and in situ hybridization analysis of the distribution of the 5-ht7 receptor in rat brain

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12 December 2020

The relaxant 5-HT receptor in the dog coronary artery smooth muscle: pharmacological resemblance to the cloned 5-ht7 receptor subtype

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12 December 2020

Antagonism of phencyclidine-induced deficits in prepulse inhibition by the putative atypical antipsychotic olanzapine

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12 December 2020

Characterization of putative 5-ht7 receptors mediating direct relaxation in Cynomolgus monkey isolated jugular vein

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12 December 2020

Functional, endogenously expressed 5-hydroxytryptamine 5-ht7 receptors in human vascular smooth muscle cells

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12 December 2020

Impact of adrenalectomy on 5-HT6 and 5-HT7 receptor gene expression in the rat hippocampus

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12 December 2020

Mediation of 5-HT-induced external carotid vasodilatation in GR 127935-pretreated vagosympathectomized dogs by the putative 5-HT7 receptor.

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12 December 2020

Blockade of phencyclidine-induced hyperlocomotion by olanzapine, clozapine and serotonin receptor subtype selective antagonists in mice

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12 December 2020

The 5-HT7 receptor: orphan found

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12 December 2020

Increase of 5-HT7 (serotonin-7) and 5-HT1A (serotonin-1A) receptor mRNA expression in rat hippocampus after adrenalectomy.

1 reference

12 December 2020

5-HT7 receptors mediate serotonergic effects on light-sensitive suprachiasmatic nucleus neurons

1 reference

12 December 2020

5-hydroxytryptamine receptor subtype messenger RNAs in human dorsal root ganglia: a polymerase chain reaction study

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12 December 2020

Do Novel Antipsychotics Have Similar Pharmacological Characteristics? A Review of the Evidence

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12 December 2020

Correlation between 5-HT7 receptor affinity and protection against sound-induced seizures in DBA/2J mice

1 reference

12 December 2020

A Test of the Predictive Validity of Animal Models of Schizophrenia Based on Phencyclidine and D-Amphetamine

1 reference

12 December 2020

(R)-3,N-Dimethyl-N-[1-methyl-3-(4-methylpiperidin-1-yl)propyl]benzenesulfonamide: The First Selective 5-HT7Receptor Antagonist

1 reference

12 December 2020

Functional characterisation of the human cloned 5-HT7 receptor (long form); antagonist profile of SB-258719

1 reference

12 December 2020

Antisense oligonucleotide-induced reduction in 5-hydroxytryptamine7 receptors in the rat hypothalamus without alteration in exploratory behaviour or neuroendocrine function

1 reference

12 December 2020

Effect of novel antipsychotic drugs on phencyclidine-induced stereotyped behaviour and social isolation in the rat social interaction test.

1 reference

12 December 2020

Involvement of the 5-HT7 receptor in craniovascular vasodilatation: potential impact in migraine.

1 reference

12 December 2020

Oxytocin modulates psychotomimetic-induced deficits in sensorimotor gating

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12 December 2020

10.1111/J.1527-3458.2002.TB00217.X

Identifiers

DOI

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12070528 AND SRC:MED&resulttype=core&format=json

10 November 2019

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12070528 AND SRC:MED&resulttype=core&format=json

10 November 2019

PubMed publication ID

12070528

1 reference