β-Lactones Inhibit N-acylethanolamine Acid Amidase by S-Acylation of the Catalytic N-Terminal Cysteine (Q34423074)

24900487

2 August 2017

title

β-Lactones Inhibit N-acylethanolamine Acid Amidase by S-Acylation of the Catalytic N-Terminal Cysteine (English)

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2 August 2017

1

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7 June 2020

Gianpiero Garau

8

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Marco Mor

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author name string

Elisa Romeo

2

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Stefano Ponzano

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Luisa Mengatto

4

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Mauro Dionisi

5

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Claudia Karacsonyi

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Fabio Bertozzi

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Glauco Tarozzo

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Angelo Reggiani

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Tiziano Bandiera

11

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Giorgio Tarzia

12

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Daniele Piomelli

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language of work or name

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6 April 2012

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24900487

ACS Medicinal Chemistry Letters

2 August 2017

published in

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volume

3

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issue

5

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page(s)

422-426

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A catalytically silent FAAH-1 variant drives anandamide transport in neurons

7 June 2020

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Synthesis and structure-activity relationships of N-(2-oxo-3-oxetanyl)amides as N-acylethanolamine-hydrolyzing acid amidase inhibitors.

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6 July 2018

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Selective N-acylethanolamine-hydrolyzing acid amidase inhibition reveals a key role for endogenous palmitoylethanolamide in inflammation.

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The FAAH inhibitor URB-597 interferes with cisplatin- and nicotine-induced vomiting in the Suncus murinus (house musk shrew)

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Characterisation of the cannabinoid receptor system in synovial tissue and fluid in patients with osteoarthritis and rheumatoid arthritis

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The fatty acid amide hydrolase inhibitor URB597 (cyclohexylcarbamic acid 3'-carbamoylbiphenyl-3-yl ester) reduces neuropathic pain after oral administration in mice

6 July 2018

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Pharmacological profile of the selective FAAH inhibitor KDS-4103 (URB597).

6 July 2018

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Antidepressant-like activity and modulation of brain monoaminergic transmission by blockade of anandamide hydrolysis

6 July 2018

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6 July 2018

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The search for the palmitoylethanolamide receptor.

6 July 2018

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Molecular characterization of N-acylethanolamine-hydrolyzing acid amidase, a novel member of the choloylglycine hydrolase family with structural and functional similarity to acid ceramidase

6 July 2018

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N-cyclohexanecarbonylpentadecylamine: a selective inhibitor of the acid amidase hydrolysing N-acylethanolamines, as a tool to distinguish acid amidase from fatty acid amide hydrolase

6 July 2018

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6 July 2018

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Appendix 5. Nomenclature for peptide fragment ions (positive ions).

6 July 2018

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6 July 2018

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27 October 2018

Identifiers

DOI

10.1021/ML300056Y

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7 June 2020

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24900487

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