Design and pharmacological characterization of VUF14480, a covalent partial agonist that interacts with cysteine 98(3.36) of the human histamine H₄ receptor. (Q34324177)

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English	Design and pharmacological characterization of VUF14480, a covalent partial agonist that interacts with cysteine 98(3.36) of the human histamine H₄ receptor.	scientific article

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22 February 2020

Design and pharmacological characterization of VUF14480, a covalent partial agonist that interacts with cysteine 98(3.36) of the human histamine H₄ receptor (English)

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Saskia Nijmeijer

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H Engelhardt

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A C van de Stolpe

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V Lusink

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M Wijtmans

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E E J Haaksma

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I J P de Esch

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K Stachurski

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H F Vischer

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R Leurs

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22 February 2020

Analysis of multiple histamine H₄ receptor compound classes uncovers Gαi protein- and β-arrestin2-biased ligands

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Ligand based design of novel histamine H₄ receptor antagonists; fragment optimization and analysis of binding kinetics

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12 December 2020

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22 February 2020

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22 February 2020

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