Orphanin FQ/nociceptin receptor binding studies (Q34040147)

30 July 2017

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title

Orphanin FQ/nociceptin receptor binding studies (English)

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30 July 2017

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Dooley CT

1

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30 July 2017

Houghten RA

series ordinal

2

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30 July 2017

publication date

1 July 2000

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30 July 2017

number of pages

12

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inferred from page(s)

published in

Peptides

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30 July 2017

volume

21

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30 July 2017

issue

7

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30 July 2017

page(s)

949-960

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Relationship between binding affinity and functional activity of nociceptin/orphanin FQ

30 July 2017

cites work

1 reference

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7 January 2021

Interaction of [3H]orphanin FQ and 125I-Tyr14-orphanin FQ with the orphanin FQ receptor: kinetics and modulation by cations and guanine nucleotides

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7 January 2021

The stereoselective kappa-opioid receptor antagonist Mr 2266 does not exhibit stereoselectivity as an antagonist at the orphan opioid (ORL1) receptor

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7 January 2021

Ligands for kappa-opioid and ORL1 receptors identified from a conformationally constrained peptide combinatorial library

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7 January 2021

Nociceptin binding sites in frog (Rana esculenta) brain membranes.

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7 January 2021

Antagonism by acetyl-RYYRIK-NH2 of G protein activation in rat brain preparations and of chronotropic effect on rat cardiomyocytes evoked by nociceptin/orphanin FQ.

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7 January 2021

Characterization of nociceptin receptors in the periphery: in vitro and in vivo studies

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7 January 2021

Molecular cloning and tissue distribution of a putative member of the rat opioid receptor gene family that is not a mu, delta or kappa opioid receptor type

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7 January 2021

Recognition and activation of the opioid receptor-like ORL 1 receptor by nociceptin, nociceptin analogs and opioids

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7 January 2021

[Phe1psi(CH2-NH)Gly2]nociceptin-(1-13)-NH2 is an agonist of the nociceptin (ORL1) receptor.

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7 January 2021

Nociceptin, a novel endogenous ligand for the ORL1 receptor, dilates isolated resistance arteries from the rat.

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7 January 2021

Molecular cloning, tissue distribution and chromosomal localization of a novel member of the opioid receptor gene family

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7 January 2021

Endogenous opioid receptor-like receptor in human neuroblastoma SK-N-SH cells: activation of inhibitory G protein and homologous desensitization

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7 January 2021

Nociceptin receptor coupling to a potassium conductance in rat locus coeruleus neurones in vitro

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7 January 2021

Orphanin FQ: receptor binding and analog structure activity relationships in rat brain

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7 January 2021

Characterization of the high affinity [3H]nociceptin binding site in membrane preparations of rat heart: correlations with the non-opioid dynorphin binding site

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7 January 2021

Cloning of a delta opioid receptor by functional expression

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7 January 2021

Nociceptin activation of the human ORL1 receptor expressed in Chinese hamster ovary cells: Functional homology with opioid receptors

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7 January 2021

125ITyr14Orphanin binding to rat brain: evidence for labelling the opioid-receptor-like 1 (ORL1)

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7 January 2021

cDNA cloning and regional distribution of a novel member of the opioid receptor family.

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7 January 2021

Address and message sequences for the nociceptin receptor: a structure-activity study of nociceptin-(1-13)-peptide amide.

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7 January 2021

A new selective antagonist of the nociceptin receptor.

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7 January 2021

Nociceptin/orphanin FQ binding increases in superficial laminae of the rat spinal cord during persistent peripheral inflammation

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Diuretic and antinatriuretic responses produced by the endogenous opioid-like peptide, nociceptin (orphanin FQ).

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

The NMDA receptor antagonist, NPC 12626, reduces the pronociceptive effects of orphanin FQ and kappa opiate antinociception in the land snail, Cepaea nemoralis.

1 reference

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7 January 2021

Discovery of the first potent and selective small molecule opioid receptor-like (ORL1) antagonist: 1-[(3R,4R)-1-cyclooctylmethyl-3- hydroxymethyl-4-piperidyl]-3-ethyl-1, 3-dihydro-2H-benzimidazol-2-one (J-113397)

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7 January 2021

The delta-opioid receptor: isolation of a cDNA by expression cloning and pharmacological characterization

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Molecular cloning of a novel G protein-coupled receptor related to the opiate receptor family

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Comparison of the structure-activity relationships of nociceptin and dynorphin A using chimeric peptides

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Functional expression, activation and desensitization of opioid receptor-like receptor ORL1 in neuroblastoma x glioma NG108-15 hybrid cells

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Presence of nociceptin (orphanin FQ) receptors in rat retina: Comparison with receptors in striatum

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Presence and characterization of nociceptin (orphanin FQ) receptor binding in adult rat and human fetal hypothalamus

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Biochemical evidence for orphanin FQ/nociceptin receptor heterogeneity in mouse brain

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Moving from the orphanin FQ receptor to an opioid receptor using four point mutations

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Isolation and structure of the endogenous agonist of opioid receptor-like ORL1 receptor

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Replacement of Gln280 by His in TM6 of the human ORL1 receptor increases affinity but reduces intrinsic activity of opioids.

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Distinct mechanisms for activation of the opioid receptor-like 1 and kappa-opioid receptors by nociceptin and dynorphin A.

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

ORL1, a novel member of the opioid receptor family. Cloning, functional expression and localization

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Nociceptin/orphanin FQ metabolism: role of aminopeptidase and endopeptidase 24.15.

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Pharmacological studies on the "orphan" opioid receptor in central and peripheral sites

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Loss of antinociception induced by naloxone benzoylhydrazone in nociceptin receptor-knockout mice.

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Primary structure and tissue distribution of the orphanin FQ precursor

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Rat central ORL-1 receptor uncouples from adenylyl cyclase during membrane preparation.

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Comparison of the effects of [Phe1psi(CH2-NH)Gly2]nociceptin(1-13)NH2 in rat brain, rat vas deferens and CHO cells expressing recombinant human nociceptin receptors

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Dissociation of affinity and efficacy in KOR-3 chimeras

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Structure-activity relationship studies on the novel neuropeptide orphanin FQ.

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Structures That Delineate Orphanin FQ and Dynorphin A Pharmacological Selectivities

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Orphanin FQ: a neuropeptide that activates an opioidlike G protein-coupled receptor.

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Sensitivity of opioid receptor-like receptor ORL1 for chemical modification on nociceptin, a naturally occurring nociceptive peptide

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Identification of opioid receptor-like (ORL1) peptide-stimulated [35S]GTP gamma S binding in rat brain.

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Nociceptin receptor binding in mouse forebrain membranes: thermodynamic characteristics and structure activity relationships

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

cDNA cloning of an orphan opiate receptor gene family member and its splice variant

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Further characterization of the ORL1 receptor-mediated inhibition of noradrenaline release in the mouse brain in vitro

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Isolation of a novel cDNA encoding a putative membrane receptor with high homology to the cloned mu, delta, and kappa opioid receptors.

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Agonistic effect of buprenorphine in a nociceptin/OFQ receptor-triggered reporter gene assay

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Orphanin FQ has an inhibitory effect on the guinea pig ileum and the mouse vas deferens

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

Identification of dynorphins as endogenous ligands for an opioid receptor-like orphan receptor

1 reference

https://api.crossref.org/works/10.1016/S0196-9781(00)00231-X

7 January 2021

10.1016/S0196-9781(00)00231-X

Identifiers

DOI

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30 July 2017

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