Development of a high-throughput fluorescence polarization assay to identify novel ligands of glutamate carboxypeptidase II (Q33957067)

30 July 2017

title

Development of a high-throughput fluorescence polarization assay to identify novel ligands of glutamate carboxypeptidase II (English)

1 reference

30 July 2017

7

Barbara Slusher

1 reference

30 July 2017

6

Camilo Rojas

1 reference

30 July 2017

5

Marigo Stathis

1 reference

30 July 2017

8

Martin G Pomper

1 reference

30 July 2017

Glenda Alquicer

1

1 reference

30 July 2017

David Sedlák

2

1 reference

30 July 2017

Youngjoo Byun

3

1 reference

30 July 2017

Jirí Pavlícek

4

1 reference

30 July 2017

Petr Bartunek

9

1 reference

30 July 2017

Cyril Barinka

10

1 reference

30 July 2017

publication date

29 June 2012

1 reference

Journal of Biomolecular Screening

30 July 2017

published in

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30 July 2017

volume

17

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30 July 2017

issue

8

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30 July 2017

page(s)

1030-1040

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Structure-activity relationships of glutamate carboxypeptidase II (GCPII) inhibitors

30 July 2017

cites work

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4112551

5 July 2018

GCPII imaging and cancer

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4112551

Glutamate in CNS neurodegeneration and cognition and its regulation by GCPII inhibition

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4112551

The role of glutamate signaling in pain processes and its regulation by GCP II inhibition

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4112551

Glutamate carboxypeptidase II: an overview of structural studies and their importance for structure-based drug design and deciphering the reaction mechanism of the enzyme

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4112551

Tissue distribution of glutamate carboxypeptidase II (GCPII) with a focus on the central and peripheral nervous system.

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4112551

Glutamate carboxypeptidase II in diagnosis and treatment of neurologic disorders and prostate cancer

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4112551

Spacer length effects on in vitro imaging and surface accessibility of fluorescent inhibitors of prostate specific membrane antigen

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4112551

Novel Substrate-Based Inhibitors of Human Glutamate Carboxypeptidase II with Enhanced Lipophilicity

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4112551

A remote arene-binding site on prostate specific membrane antigen revealed by antibody-recruiting small molecules

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4112551

Interactions between human glutamate carboxypeptidase II and urea-based inhibitors: structural characterization

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4112551

Progress in the discovery and development of glutamate carboxypeptidase II inhibitors

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4112551

Substrate specificity of prostate-specific membrane antigen

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4112551

Biochemical characterization of human glutamate carboxypeptidase III

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4112551

Expression of glutamate carboxypeptidase II in human brain

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4112551

Technology insight: monoclonal antibody imaging of prostate cancer

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4112551

NAAG peptidase inhibitors and their potential for diagnosis and therapy

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4112551

A general framework for development and data analysis of competitive high-throughput screens for small-molecule inhibitors of protein-protein interactions by fluorescence polarization

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4112551

Amino acids at the N- and C-termini of human glutamate carboxypeptidase II are required for enzymatic activity and proper folding.

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4112551

Improved statistical methods for hit selection in high-throughput screening

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4112551

Fluorescence polarization: past, present and future

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4112551

Kinetics and inhibition of glutamate carboxypeptidase II using a microplate assay

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4112551

Design of remarkably simple, yet potent urea-based inhibitors of glutamate carboxypeptidase II (NAALADase)

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4112551

A Simple Statistical Parameter for Use in Evaluation and Validation of High Throughput Screening Assays

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4112551

Hydrolysis of the brain dipeptide N-acetyl-L-aspartyl-L-glutamate. Identification and characterization of a novel N-acetylated alpha-linked acidic dipeptidase activity from rat brain.

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4112551

Radiohalogenated prostate-specific membrane antigen (PSMA)-based ureas as imaging agents for prostate cancer

5 July 2018

1 reference

Crossref

https://api.crossref.org/works/10.1177/1087057112451924

High-performance liquid chromatography method for detecting prostate-specific membrane antigen activity

21 January 2018

1 reference

Crossref

https://api.crossref.org/works/10.1177/1087057112451924

Substrate specificity, inhibition and enzymological analysis of recombinant human glutamate carboxypeptidase II.

21 January 2018

1 reference

Crossref

https://api.crossref.org/works/10.1177/1087057112451924

Selective inhibition of NAALADase, which converts NAAG to glutamate, reduces ischemic brain injury

21 January 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/22751730

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Tissue expression and enzymologic characterization of human prostate specific membrane antigen and its rat and pig orthologs

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/22751730

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

A dual-monoclonal sandwich assay for prostate-specific membrane antigen: levels in tissues, seminal fluid and urine

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/22751730

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1177/1087057112451924

1 reference

30 July 2017

1 reference

30 July 2017

1 reference