Development and validation of a high-content screening assay to identify inhibitors of cytoplasmic dynein-mediated transport of glucocorticoid receptor to the nucleus (Q30416877)

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English	Development and validation of a high-content screening assay to identify inhibitors of cytoplasmic dynein-mediated transport of glucocorticoid receptor to the nucleus	scientific article

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scholarly article

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Europe PubMed Central

PMC publication ID

13 August 2017

Development and validation of a high-content screening assay to identify inhibitors of cytoplasmic dynein-mediated transport of glucocorticoid receptor to the nucleus (English)

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Europe PubMed Central

PMC publication ID

13 August 2017

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5

object named as

John S Lazo

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

4

object named as

Tong Ying Shun

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Europe PubMed Central

PMC publication ID

13 August 2017

Sunita N Shinde

2

object named as

Sunita N Shinde

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Europe PubMed Central

PMC publication ID

13 August 2017

author name string

Paul A Johnston

1

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Europe PubMed Central

PMC publication ID

13 August 2017

Yun Hua

3

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Europe PubMed Central

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13 August 2017

Billy W Day

6

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Europe PubMed Central

PMC publication ID

13 August 2017

publication date

25 July 2012

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Europe PubMed Central

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13 August 2017

Assay and Drug Development Technologies

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Europe PubMed Central

PMC publication ID

13 August 2017

10

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Europe PubMed Central

PMC publication ID

13 August 2017

5

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

432-456

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Europe PubMed Central

PMC publication ID

13 August 2017

Characterization of inhibitors of glucocorticoid receptor nuclear translocation: a model of cytoplasmic dynein-mediated cargo transport.

1 reference

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Mechanisms generating diversity in glucocorticoid receptor signaling.

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Glucocorticoid signaling in the cell. Expanding clinical implications to complex human behavioral and somatic disorders

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Kinesin superfamily motor proteins and intracellular transport

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Nuclear import of the glucocorticoid receptor-hsp90 complex through the nuclear pore complex is mediated by its interaction with Nup62 and importin beta

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High-throughput automated confocal microscopy imaging screen of a kinase-focused library to identify p38 mitogen-activated protein kinase inhibitors using the GE InCell 3000 analyzer

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Emerging roles for myosin II and cytoplasmic dynein in migrating neurons and growth cones

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The glucocorticoid responses are shaped by molecular chaperones

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Geldanamycin, an inhibitor of Hsp90, blocks cytoplasmic retention of progesterone receptors and glucocorticoid receptors via their respective ligand binding domains

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International Union of Pharmacology. LXV. The pharmacology and classification of the nuclear receptor superfamily: glucocorticoid, mineralocorticoid, progesterone, and androgen receptors

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Assay development and case history of a 32K-biased library high-content MK2-EGFP translocation screen to identify p38 mitogen-activated protein kinase inhibitors on the ArrayScan 3.1 imaging platform

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Generation and characterization of a stable MK2-EGFP cell line and subsequent development of a high-content imaging assay on the Cellomics ArrayScan platform to screen for p38 mitogen-activated protein kinase inhibitors

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Autoinhibitory and other autoregulatory elements within the dynein motor domain

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Synthesis and biological evaluation of purealin and analogues as cytoplasmic dynein heavy chain inhibitors.

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Microtubule-interfering activity of parthenolide

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10.1089/ADT.2012.456

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

PMC publication ID

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

PubMed publication ID

1 reference

Europe PubMed Central

PMC publication ID

13 August 2017

ResearchGate publication ID

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