Synthesis, antitubercular activity and mechanism of resistance of highly effective thiacetazone analogues (Q28484824)

1

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Derek Craig

2

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Rosa Milagros Corrales

3

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Emilie Vialla

4

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Laila Gannoun-Zaki

Creative Commons Attribution 4.0 International

5

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language of work or name

English

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publication date

2013

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published in

PLOS One

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volume

8

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issue

1

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page(s)

e53162

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copyright license

start time

3 January 2013

1 reference

April 2022 Public Data File from Crossref

copyright status

copyrighted

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cites work

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Negative regulation by Ser/Thr phosphorylation of HadAB and HadBC dehydratases from Mycobacterium tuberculosis type II fatty acid synthase system

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Preclinical pharmacokinetics of KBF611, a new antituberculosis agent in mice and rabbits, and comparison with thiacetazone

21 January 2018

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Thiacetazone--use with care

21 January 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/23301038

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

1 reference

https://pubmed.ncbi.nlm.nih.gov/23301038

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Mutations in the essential FAS II β-hydroxyacyl ACP dehydratase complex confer resistance to thiacetazone in Mycobacterium tuberculosis and Mycobacterium kansasii

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/23301038

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1371/JOURNAL.PONE.0053162

1 reference

ADS bibcode

2013PLoSO...853162C

0 references

1 reference

1 reference

PubMed publication ID

23301038

1 reference