BAY36-7620: a potent non-competitive mGlu1 receptor antagonist with inverse agonist activity (Q28362867)

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6 November 2019

title

BAY36-7620: a potent non-competitive mGlu1 receptor antagonist with inverse agonist activity (English)

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11

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author name string

Carroll FY

1

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6 November 2019

Stolle A

2

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Beart PM

3

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Voerste A

4

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Brabet I

5

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Mauler F

6

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Joly C

7

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Antonicek H

8

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Bockaert J

9

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Müller T

10

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Prézeau L

12

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language of work or name

English

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publication date

1 May 2001

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6 November 2019

published in

Molecular Pharmacology

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volume

59

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issue

5

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6 November 2019

page(s)

965-973

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Structural basis of glutamate recognition by a dimeric metabotropic glutamate receptor

6 November 2019

cites work

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Measurement of protein using bicinchoninic acid

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Constitutive G(i2)-dependent activation of adenylyl cyclase type II by the 5-HT1A receptor. Inhibition by anxiolytic partial agonists

29 September 2017

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29 September 2017

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New perspectives for the development of selective metabotropic glutamate receptor ligands.

29 September 2017

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Comparative effect of L-CCG-I, DCG-IV and gamma-carboxy-L-glutamate on all cloned metabotropic glutamate receptor subtypes.

29 September 2017

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Expression and purification of the extracellular ligand binding region of metabotropic glutamate receptor subtype 1.

29 September 2017

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The G protein-coupling profile of metabotropic glutamate receptors, as determined with exogenous G proteins, is independent of their ligand recognition domain

29 September 2017

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Substitution of three amino acids switches receptor specificity of Gq alpha to that of Gi alpha

29 September 2017

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The ligand-binding domain in metabotropic glutamate receptors is related to bacterial periplasmic binding proteins

29 September 2017

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Constitutive activity of receptors coupled to guanine nucleotide regulatory proteins

29 September 2017

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A mutation-induced activated state of the beta 2-adrenergic receptor. Extending the ternary complex model

29 September 2017

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29 September 2017

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Molecular, functional, and pharmacological characterization of the metabotropic glutamate receptor type 5 splice variants: comparison with mGluR1.

29 September 2017

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Regions of the alpha 1-adrenergic receptor involved in coupling to phosphatidylinositol hydrolysis and enhanced sensitivity of biological function

29 September 2017

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29 September 2017

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29 September 2017

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Pharmacological characterization of metabotropic glutamate receptors in several types of brain cells in primary cultures.

27 November 2018

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The non-competitive antagonists 2-methyl-6-(phenylethynyl)pyridine and 7-hydroxyiminocyclopropan[b]chromen-1a-carboxylic acid ethyl ester interact with overlapping binding pockets in the transmembrane region of group I metabotropic glutamate recepto

27 November 2018

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12 December 2020

Reversible and non-competitive antagonist profile of CPCCOEt at the human type 1alpha metabotropic glutamate receptor

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12 December 2020

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12 December 2020

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12 December 2020

Identifiers

DOI

10.1124/MOL.59.5.965

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11306677 AND SRC:MED&resulttype=core&format=json

6 November 2019

1290425

1 reference

Consolidated OpenCitations Corpus – April 2017

Consolidated OpenCitations Corpus – April 2017

2 references

1290425

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:11306677 AND SRC:MED&resulttype=core&format=json

6 November 2019

PubMed publication ID

11306677

2 references

Consolidated OpenCitations Corpus – April 2017

1290425