Structural basis of inhibition of Mycobacterium tuberculosis DprE1 by benzothiazinone inhibitors (Q27681391)

8

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Luke J Alderwick

object named as

Luke J Alderwick

7

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Gurdyal Besra

object named as

Gurdyal S Besra

9

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author name string

Sarah M Batt

1

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Talat Jabeen

2

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Veemal Bhowruth

3

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Lee Quill

4

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Peter A Lund

5

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Lothar Eggeling

Proceedings of the National Academy of Sciences of the United States of America

6

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language of work or name

English

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publication date

10 July 2012

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published in

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volume

109

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issue

28

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page(s)

11354-9

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cites work

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Crystal structures and inhibitor binding in the octameric flavoenzyme vanillyl-alcohol oxidase: the shape of the active-site cavity controls substrate specificity

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Methods used in the structure determination of bovine mitochondrial F1 ATPase

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Characteristics and treatment outcomes of patients with MDR and XDR tuberculosis in a TB referral hospital in Beijing: a 13-year experience

20 March 2017

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Biochemical characterization of the Mycobacterium tuberculosis phosphoribosyl-1-pyrophosphate synthetase

20 March 2017

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High content screening identifies decaprenyl-phosphoribose 2' epimerase as a target for intracellular antimycobacterial inhibitors

20 March 2017

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Benzothiazinones kill Mycobacterium tuberculosis by blocking arabinan synthesis

20 March 2017

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Decaprenylphosphoryl arabinofuranose, the donor of the D-arabinofuranosyl residues of mycobacterial arabinan, is formed via a two-step epimerization of decaprenylphosphoryl ribose

20 March 2017

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Genes required for mycobacterial growth defined by high density mutagenesis

20 March 2017

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Benzothiazinones are suicide inhibitors of mycobacterial decaprenylphosphoryl-β-D-ribofuranose 2'-oxidase DprE1.

20 March 2017

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Decaprenylphosphoryl-β-D-ribose 2'-epimerase from Mycobacterium tuberculosis is a magic drug target

29 September 2017

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Multidrug-resistant and extensively drug-resistant tuberculosis: a threat to global control of tuberculosis

29 September 2017

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Clinical isolates of Mycobacterium tuberculosis in four European hospitals are uniformly susceptible to benzothiazinones

29 September 2017

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The growing VAO flavoprotein family.

29 September 2017

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Structure, function and biosynthesis of the Mycobacterium tuberculosis cell wall: arabinogalactan and lipoarabinomannan assembly with a view to discovering new drug targets.

29 September 2017

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Benzothiazinones: prodrugs that covalently modify the decaprenylphosphoryl-β-D-ribose 2'-epimerase DprE1 of Mycobacterium tuberculosis

29 September 2017

1 reference

Crossref

https://api.crossref.org/works/10.1073/PNAS.1205735109

Totally Drug-Resistant Tuberculosis in India

21 January 2018

1 reference

Crossref

https://api.crossref.org/works/10.1073/PNAS.1205735109

Phasing in the presence of severe site-specific radiation damage through dose-dependent modelling of heavy atoms

21 January 2018

1 reference

Crossref

https://api.crossref.org/works/10.1073/PNAS.1205735109

Polyprenylphosphate-pentoses in mycobacteria are synthesized from 5-phosphoribose pyrophosphate

21 January 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/22733761

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1073/PNAS.1205735109

1 reference

ADS bibcode

2012PNAS..10911354B

0 references

1 reference

1 reference

PubMed publication ID

22733761

1 reference