A surface on the androgen receptor that allosterically regulates coactivator binding (Q27648698)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17911242 AND SRC:MED&resulttype=core&format=json

8 January 2020

title

A surface on the androgen receptor that allosterically regulates coactivator binding (English)

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17911242 AND SRC:MED&resulttype=core&format=json

Correction for Estébanez-Perpiñá et al., A surface on the androgen receptor that allosterically regulates coactivator binding

8 January 2020

corrigendum / erratum

0 references

author

Eva Estébanez-Perpiñá

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17911242 AND SRC:MED&resulttype=core&format=json

8 January 2020

R. Kiplin Guy

10

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17911242 AND SRC:MED&resulttype=core&format=json

8 January 2020

Leggy A Arnold

2

0 references

Robert Fletterick

12

object named as

Robert J Fletterick

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17911242 AND SRC:MED&resulttype=core&format=json

8 January 2020

11

Paul Webb

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17911242 AND SRC:MED&resulttype=core&format=json

8 January 2020

5

Ellena Mar

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17911242 AND SRC:MED&resulttype=core&format=json

8 January 2020

author name string

Phuong Nguyen

3

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17911242 AND SRC:MED&resulttype=core&format=json

8 January 2020

Edson Delgado Rodrigues

4

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17911242 AND SRC:MED&resulttype=core&format=json

8 January 2020

Raynard Bateman

6

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17911242 AND SRC:MED&resulttype=core&format=json

8 January 2020

Peter Pallai

7

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17911242 AND SRC:MED&resulttype=core&format=json

8 January 2020

Kevan M Shokat

8

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17911242 AND SRC:MED&resulttype=core&format=json

8 January 2020

John D Baxter

9

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17911242 AND SRC:MED&resulttype=core&format=json

8 January 2020

language of work or name

English

0 references

publication date

2 October 2007

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17911242 AND SRC:MED&resulttype=core&format=json

Proceedings of the National Academy of Sciences of the United States of America

8 January 2020

published in

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17911242 AND SRC:MED&resulttype=core&format=json

8 January 2020

volume

104

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17911242 AND SRC:MED&resulttype=core&format=json

8 January 2020

issue

41

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17911242 AND SRC:MED&resulttype=core&format=json

8 January 2020

page(s)

16074-16079

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17911242 AND SRC:MED&resulttype=core&format=json

The molecular mechanisms of coactivator utilization in ligand-dependent transactivation by the androgen receptor

8 January 2020

cites work

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

Recognition and accommodation at the androgen receptor coactivator binding interface

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

In vivo activation of the p53 pathway by small-molecule antagonists of MDM2

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

Ligand selectivity by seeking hydrophobicity in thyroid hormone receptor

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

Crystallographic comparison of the estrogen and progesterone receptor's ligand binding domains

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

Nuclear-receptor ligands and ligand-binding domains

20 March 2017

2 references

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

20 March 2017

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

Androgen receptor-cofactor interactions as targets for new drug discovery

7 April 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

Sensors and signals: a coactivator/corepressor/epigenetic code for integrating signal-dependent programs of transcriptional response

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

Androgen receptor in prostate cancer

7 April 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

Small-molecule inhibitors of protein-protein interactions: progressing towards the dream

7 April 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

The nuclear receptor LXR is a glucose sensor

7 April 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

Treatment of Postmenopausal Breast Cancer with Selective Estrogen Receptor Modulators (SERMs).

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

A second binding site for hydroxytamoxifen within the coactivator-binding groove of estrogen receptor beta

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

The expanding cosmos of nuclear receptor coactivators

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

Molecular regulation of androgen action in prostate cancer

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

Biology of progressive, castration-resistant prostate cancer: directed therapies targeting the androgen-receptor signaling axis

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

Development of peptide antagonists for the androgen receptor using combinatorial peptide phage display

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

Ligand control of coregulator recruitment to nuclear receptors

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

Signature of the oligomeric behaviour of nuclear receptors at the sequence and structural level

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

Finding specificity within a conserved interaction site

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

Modulation of protein-protein interactions with small organic molecules

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

The development of COX2 inhibitors

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

Androgen receptor mutations and androgen insensitivity

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

Progress toward the development of agents to modulate the cell cycle

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

The NH(2)-terminal and carboxyl-terminal interaction in the human androgen receptor

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

Structure-based design and synthesis of a thyroid hormone receptor (TR) antagonist.

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

Mutations at the boundary of the hinge and ligand binding domain of the androgen receptor confer increased transactivation function

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

Discovering novel ligands for macromolecules using X-ray crystallographic screening

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

Human androgen receptor mutation disrupts ternary interactions between ligand, receptor domains, and the coactivator TIF2 (transcription intermediary factor 2).

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

Discovery of small molecule inhibitors of the interaction of the thyroid hormone receptor with transcriptional coregulators

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

Hormone-dependent coactivator binding to a hydrophobic cleft on nuclear receptors

2 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

Identification of amino acids in the tau 2-region of the mouse glucocorticoid receptor that contribute to hormone binding and transcriptional activation

2 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

Design, synthesis, and in vitro biological evaluation of small molecule inhibitors of estrogen receptor alpha coactivator binding

2 June 2018

1 reference

Crossref

https://api.crossref.org/works/10.1073/PNAS.0708036104

Novel molecular defects in the androgen receptor gene of Mexican patients with androgen insensitivity

21 January 2018

1 reference

Crossref

https://api.crossref.org/works/10.1073/PNAS.0708036104

Dihydrotestosterone (DHT) modulates the ability of NSAIDs to induce apoptosis of prostate cancer cells

21 January 2018

1 reference

Crossref

https://api.crossref.org/works/10.1073/PNAS.0708036104

Functional analysis of 44 mutant androgen receptors from human prostate cancer.

21 January 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1999396

Drug discovery at signaling interfaces

27 November 2018

1 reference

12 December 2020

Structural basis for androgen receptor interdomain and coactivator interactions suggests a transition in nuclear receptor activation function dominance

1 reference

12 December 2020

A high-throughput screening method to identify small molecule inhibitors of thyroid hormone receptor coactivator binding

1 reference

12 December 2020

Collocation of androgen receptor gene mutations in prostate cancer

1 reference

12 December 2020

Identifiers

DOI

10.1073/PNAS.0708036104

2 references

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17911242 AND SRC:MED&resulttype=core&format=json

8 January 2020

ADS bibcode

2007PNAS..10416074E

0 references

1 reference

2 references

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17911242 AND SRC:MED&resulttype=core&format=json

8 January 2020

PubMed publication ID

17911242

2 references